N-substituted Piperazinopyridylsteroid Derivatives as Abiraterone Analogues Inhibit Growth and Induce Pro-apoptosis in Human Hormone-independent Prostate Cancer Cell Lines

Aromatase: The Enzyme and Its Inhibition

(2012) Lee Banting et al.   Anti-Cancer Agents in Medicinal Chemistry

17α-Hydroxylase/17,20-Lyase (P450 ) Inhibitors in the Treatment of Prostate Cancer: A Review

(2012) Caroline Owen   Anti-Cancer Agents in Medicinal Chemistry

The evolving paradigm of second-line hormonal therapy options for castration-resistant prostate cancer

(2012) Kevin D. Courtney et al.   CURRENT OPINION IN ONCOLOGY

Aromatase inhibitors and breast cancer prevention

(2012) Jennifer Keating Litton et al.   EXPERT OPINION ON PHARMACOTHERAPY

A new investigation for some steroidal derivatives as anti-Alzheimer agents

(2012) Mohamed M. Abdalla et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Heterocyclizations of pregnenolone: Novel synthesis of thiosemicarbazone, thiophene, thiazole, thieno[2,3-b]pyridine derivatives and their cytotoxicity evaluations

(2012) Rafat M. Mohareb et al.   STEROIDS

Aromatase, aromatase inhibitors, and breast cancer

(2011) Saranya Chumsri et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

α-Chaconine Inhibits Angiogenesis in Vitro by Reducing Matrix Metalloproteinase-2

(2010) Ming-Kun Lu et al.   BIOLOGICAL & PHARMACEUTICAL BULLETIN

α-Solanine Inhibits Human Melanoma Cell Migration and Invasion by Reducing Matrix Metalloproteinase-2/9 Activities

(2010) Ming-Kun Lu et al.   BIOLOGICAL & PHARMACEUTICAL BULLETIN

VMY-1-103, a dansylated analog of purvalanol B, induces caspase-3-dependent apoptosis in LNCaP prostate cancer cells

(2010) Lymor Ringer et al.   CANCER BIOLOGY & THERAPY

Evidence of Limited Contributions for Intratumoral Steroidogenesis in Prostate Cancer

(2010) J. Hofland et al.   CANCER RESEARCH

Molecular Modeling on Inhibitor Complexes and Active-Site Dynamics of Cytochrome P450 C17, a Target for Prostate Cancer Therapy

(2010) Shozeb M. Haider et al.   JOURNAL OF MOLECULAR BIOLOGY

CYP17 inhibitors for prostate cancer therapy

(2010) Tadas S. Vasaitis et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Chlorotrimethylsilane-promoted one-pot synthesis of steroidal[17,16-d]pyrimidines

(2010) Cunde Wang et al.   STEROIDS

The Antifungal Activity of Sarcococca saligna Ethanol Extract and its Combination Effect with Fluconazole against Different Resistant Aspergillus Species

(2009) Kamyar Mollazadeh Moghaddam et al.   APPLIED BIOCHEMISTRY AND BIOTECHNOLOGY

Synthesis and pharmacological evaluation of new arylpiperazines N-{4-[4-(aryl) piperazine-1-yl]-phenyl}-amine derivatives: Putative role of 5-HT1A receptors

(2009) Manisha Khatri et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Tissue-Selective Regulation of Aromatase Expression by Calcitriol: Implications for Breast Cancer Therapy

(2009) Aruna V. Krishnan et al.   ENDOCRINOLOGY

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

(2009) Garrett M. Morris et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY

Role of Bax in quercetin-induced apoptosis in human prostate cancer cells

(2008) Dae-Hee Lee et al.   BIOCHEMICAL PHARMACOLOGY

New lithocholic and chenodeoxycholic piperazinylcarboxamides with antiproliferative and pro-apoptotic effects on human cancer cell lines

(2008) Laïla El Kihel et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Paradoxical effect of 1-(1-naphthylmethyl)-piperazine on resistance to tetracyclines in multidrug-resistant Acinetobacter baumannii

(2008) D. C. Bean et al.   JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY

Synthesis and Biological Evaluation of 2-Amino-3-(4-Chlorobenzoyl)-4-[N-(Substituted) Piperazin-1-yl]Thiophenes as Potent Allosteric Enhancers of the A1Adenosine Receptor

(2008) Romeo Romagnoli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Microwave promoted one-pot synthesis of novel A-ring fused steroidal dehydropiperazines

(2008) Moyurima Borthakur et al.   STEROIDS