GPBA: a GPCR for bile acids and an emerging therapeutic target for disorders of digestion and sensation
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Title
GPBA: a GPCR for bile acids and an emerging therapeutic target for disorders of digestion and sensation
Authors
Keywords
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Journal
BRITISH JOURNAL OF PHARMACOLOGY
Volume 171, Issue 5, Pages 1156-1166
Publisher
Wiley
Online
2013-10-12
DOI
10.1111/bph.12426
References
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Related references
Note: Only part of the references are listed.- The Concise Guide to PHARMACOLOGY 2013/14: G Protein-Coupled Receptors
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- Weight Loss Induced by Roux-en-Y Gastric Bypass But Not Laparoscopic Adjustable Gastric Banding Increases Circulating Bile Acids
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- TGR5 potentiates GLP-1 secretion in response to anionic exchange resins
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- TGR5 Activation Inhibits Atherosclerosis by Reducing Macrophage Inflammation and Lipid Loading
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- TGR5 Sequence Variation in Primary Sclerosing Cholangitis
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- TGR5 in the Biliary Tree
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- The G-Protein-coupled bile acid receptor, Gpbar1 (TGR5), negatively regulates hepatic inflammatory response through antagonizing nuclear factor kappa light-chain enhancer of activated B cells (NF-κB) in mice
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- The G Protein-Coupled Bile Acid Receptor, TGR5, Stimulates Gallbladder Filling
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- Association of bile acid receptor TGR5 variation and transit in health and lower functional gastrointestinal disorders
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- The Bile Acid Receptor GPBAR-1 (TGR5) Modulates Integrity of Intestinal Barrier and Immune Response to Experimental Colitis
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- The Itch of Liver Disease
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- Hydrophobic bile salts inhibit gallbladder smooth muscle function via stimulation of GPBAR1 receptors and activation of KATPchannels
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- Serum bile acid along with plasma incretins and serum high–molecular weight adiponectin levels are increased after bariatric surgery
- (2009) Hiroshi Nakatani et al. METABOLISM-CLINICAL AND EXPERIMENTAL
- Serum Bile Acids Are Higher in Humans With Prior Gastric Bypass: Potential Contribution to Improved Glucose and Lipid Metabolism
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- Courvoisier’s Gallbladder: Law or Sign?
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- Expression and function of the bile acid receptor TGR5 in Kupffer cells
- (2008) Verena Keitel et al. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
- Bile Acids: Chemistry, Pathochemistry, Biology, Pathobiology, and Therapeutics
- (2008) A. F. Hofmann et al. CELLULAR AND MOLECULAR LIFE SCIENCES
- Novel Potent and Selective Bile Acid Derivatives as TGR5 Agonists: Biological Screening, Structure−Activity Relationships, and Molecular Modeling Studies
- (2008) Hiroyuki Sato et al. JOURNAL OF MEDICINAL CHEMISTRY
- Metabolic profiling of the human response to a glucose challenge reveals distinct axes of insulin sensitivity
- (2008) Oded Shaham et al. Molecular Systems Biology
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