Deciphering µ-opioid receptor phosphorylation and dephosphorylation in HEK293 cells

Agonist-selective patterns of µ-opioid receptor phosphorylation revealed by phosphosite-specific antibodies

(2011) Christian Doll et al.   BRITISH JOURNAL OF PHARMACOLOGY

Rapid Dephosphorylation of G Protein-coupled Receptors by Protein Phosphatase 1β Is Required for Termination of β-Arrestin-dependent Signaling

(2011) Florian Pöll et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Agonist-directed Interactions with Specific β-Arrestins Determine μ-Opioid Receptor Trafficking, Ubiquitination, and Dephosphorylation

(2011) Chad E. Groer et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Analgesic Tolerance to High-Efficacy Agonists But Not to Morphine Is Diminished in Phosphorylation-Deficient S375A  -Opioid Receptor Knock-In Mice

(2011) G. Grecksch et al.   JOURNAL OF NEUROSCIENCE

Functional Selectivity at the  -Opioid Receptor: Implications for Understanding Opioid Analgesia and Tolerance

(2011) K. M. Raehal et al.   PHARMACOLOGICAL REVIEWS

Quantitative Encoding of the Effect of a Partial Agonist on Individual Opioid Receptors by Multisite Phosphorylation and Threshold Detection

(2011) E. K. Lau et al.   Science Signaling

Guidelines for reporting experiments involving animals: the ARRIVE guidelines

(2010) JC McGrath et al.   BRITISH JOURNAL OF PHARMACOLOGY

Animal research: Reporting in vivo experiments: The ARRIVE guidelines

(2010) Carol Kilkenny et al.   BRITISH JOURNAL OF PHARMACOLOGY

Agonist-dependent μ-opioid receptor signaling can lead to heterologous desensitization

(2010) Ji Chu et al.   CELLULAR SIGNALLING

Pasireotide and Octreotide Stimulate Distinct Patterns of sst2ASomatostatin Receptor Phosphorylation

(2010) Florian Pöll et al.   MOLECULAR ENDOCRINOLOGY

 -Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization

(2010) J. McPherson et al.   MOLECULAR PHARMACOLOGY

UMB-3, a novel rabbit monoclonal antibody, for assessing μ-opioid receptor expression in mouse, rat and human formalin-fixed and paraffin-embedded tissues

(2010) Amelie Lupp et al.   REGULATORY PEPTIDES

Involvement of PKCα and G-protein-coupled receptor kinase 2 in agonist-selective desensitization of µ-opioid receptors in mature brain neurons

(2009) CP Bailey et al.   BRITISH JOURNAL OF PHARMACOLOGY

The Effect of Protein Kinase C and G Protein-Coupled Receptor Kinase Inhibition on Tolerance Induced by  -Opioid Agonists of Different Efficacy

(2009) L. C. Hull et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

From Promiscuity to Precision: Protein Phosphatases Get a Makeover

(2009) David M. Virshup et al.   MOLECULAR CELL

Selective engagement of G protein coupled receptor kinases (GRKs) encodes distinct functions of biased ligands

(2009) D. A. Zidar et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Morphine-induced μ-opioid receptor rapid desensitization is independent of receptor phosphorylation and β-arrestins

(2008) Ji Chu et al.   CELLULAR SIGNALLING

Differential Effects of Octreotide and Pasireotide on Somatostatin Receptor Internalization and Traffickingin Vitro

(2008) Sarah Lesche et al.   JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM

Differential Activation and Trafficking of  -Opioid Receptors in Brain Slices

(2008) S. Arttamangkul et al.   MOLECULAR PHARMACOLOGY

Role of receptor internalization in opioid tolerance and dependence

(2007) Thomas Koch et al.   PHARMACOLOGY & THERAPEUTICS