Pharmacokinetic and pharmacodynamic profiling of a P2X7 receptor allosteric modulator GSK1482160 in healthy human subjects

Efficacy and Safety of CE-224,535, an Antagonist of P2X7 Receptor, in Treatment of Patients with Rheumatoid Arthritis Inadequately Controlled by Methotrexate

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Guide to Receptors and Channels (GRAC), 5th edition

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Non-invasive imaging in experimental medicine for drug development

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Seizure suppression and neuroprotection by targeting the purinergic P2X7 receptor during status epilepticus in mice

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P2X7 receptor blockade prevents ATP excitotoxicity in neurons and reduces brain damage after ischemia

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Cloning and pharmacological characterization of the dog P2X7 receptor

(2009) S Roman et al.   BRITISH JOURNAL OF PHARMACOLOGY

Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders

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