Synthesis of Bioactive Natural Products as Protein Inhibitors

Synthesis and cytotoxicity of the depsipeptides analogues of callipeltin B

(2011) Mari Kikuchi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of tokaramide A, a cysteine protease inhibitor from marine sponge Theonella aff. mirabilis

(2011) Hiroyuki Konno et al.   TETRAHEDRON

Solid phase total synthesis of callipeltin E isolated from marine sponge Latrunculia sp.

(2011) Mari Kikuchi et al.   TETRAHEDRON LETTERS

Synthesis of solamin type mono-THF acetogenins using cross-metathesis

(2010) Hiroyuki Konno et al.   TETRAHEDRON

Synthetic Studies on Callipeltins: Stereoselective Syntheses of (3S,4R)-3,4-Dimethyl-L-pyroglutamic Acid and Fmoc-D-allothreonine from Serine Derivatives

(2009) Hiroyuki Konno et al.   HETEROCYCLES

Evaluation of peptide-aldehyde inhibitors using R188I mutant of SARS 3CL protease as a proteolysis-resistant mutant

(2008) Kenichi Akaji et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Total synthesis of cis-solamin A, a mono-tetrahydrofuran acetogenin isolated from Annona muricata

(2007) Hiroyuki Konno et al.   TETRAHEDRON LETTERS