Bisubstrate UDP–peptide conjugates as human O-GlcNAc transferase inhibitors

O-GlcNAcylation of TAB1 modulates TAK1-mediated cytokine release

(2012) Shalini Pathak et al.   EMBO JOURNAL

Structural snapshots of the reaction coordinate for O-GlcNAc transferase

(2012) Michael B Lazarus et al.   Nature Chemical Biology

O-GlcNAc transferase invokes nucleotide sugar pyrophosphate participation in catalysis

(2012) Marianne Schimpl et al.   Nature Chemical Biology

Cell-penetrating peptides: breaking through to the other side

(2012) Erez Koren et al.   TRENDS IN MOLECULAR MEDICINE

Development of a universal glycosyltransferase assay amenable to high-throughput formats

(2011) Hyun Soo Lee et al.   ANALYTICAL BIOCHEMISTRY

A Concise Synthesis of the HCV Protease Inhibitor BILN 2061 and Its P3 Modified Analogs

(2011) Dejun Liu et al.   CHINESE JOURNAL OF CHEMISTRY

A neutral diphosphate mimic crosslinks the active site of human O-GlcNAc transferase

(2011) Jiaoyang Jiang et al.   Nature Chemical Biology

Hijacking a biosynthetic pathway yields a glycosyltransferase inhibitor within cells

(2011) Tracey M Gloster et al.   Nature Chemical Biology

Substrate and product analogues as human O-GlcNAc transferase inhibitors

(2010) Helge C. Dorfmueller et al.   AMINO ACIDS

Increasing O-GlcNAc levels: An overview of small-molecule inhibitors of O-GlcNAcase

(2009) Matthew S. Macauley et al.   BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS

Bisubstrate Inhibitors of Protein Kinases: from Principle to Practical Applications

(2009) Darja Lavogina et al.   ChemMedChem

Bisubstrate Analogues as Glycosyltransferase Inhibitors

(2009) Masayuki Izumi et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Turn-On Fluorescence Sensing of Nucleoside Polyphosphates Using a Xanthene-Based Zn(II) Complex Chemosensor

(2008) Akio Ojida et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cell-penetrating peptides as delivery vehicles for biology and medicine

(2008) Kelly M. Stewart et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A Versatile One-Pot Procedure to Phosphate Monoesters and Pyrophosphates Using Di(p-methoxybenzyl)-N,N-diisopropylphosphoramidite

(2008) Gerbrand J. van der Heden van Noort et al.   ORGANIC LETTERS