Enantiomer Selective Glucuronidation of the Non-Steroidal Pure Anti-Androgen Bicalutamide by Human Liver and Kidney: Role of the Human UDP-Glucuronosyltransferase (UGT)1A9 Enzyme

Sorafenib Is an Inhibitor of UGT1A1 but Is Metabolized by UGT1A9: Implications of Genetic Variants on Pharmacokinetics and Hyperbilirubinemia

(2012) C. J. Peer et al.   CLINICAL CANCER RESEARCH

Method for predicting human intestinal first-pass metabolism of UGT substrate compounds

(2012) Takako Furukawa et al.   XENOBIOTICA

Quantification of Human Uridine-Diphosphate Glucuronosyl Transferase 1A Isoforms in Liver, Intestine, and Kidney Using Nanobore Liquid Chromatography–Tandem Mass Spectrometry

(2011) David E. Harbourt et al.   ANALYTICAL CHEMISTRY

Characterizing the effect of UDP-glucuronosyltransferase (UGT) 2B7 and UGT1A9 genetic polymorphisms on enantioselective glucuronidation of flurbiprofen

(2011) Haina Wang et al.   BIOCHEMICAL PHARMACOLOGY

A phase II study of sorafenib in combination with bicalutamide in patients with chemotherapy-naive castration resistant prostate cancer

(2011) Emma K. Beardsley et al.   INVESTIGATIONAL NEW DRUGS

Renal UDP-glucuronosyltransferases and the glucuronidation of xenobiotics and endogenous mediators

(2010) Kathleen M. Knights et al.   DRUG METABOLISM REVIEWS

Quantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human Livers

(2009) T. Izukawa et al.   DRUG METABOLISM AND DISPOSITION

Glucuronidation of the Antiretroviral Drug Efavirenz by UGT2B7 and an in Vitro Investigation of Drug-Drug Interaction with Zidovudine

(2009) A.-S. Belanger et al.   DRUG METABOLISM AND DISPOSITION

UGT genomic diversity: beyond gene duplication

(2009) Chantal Guillemette et al.   DRUG METABOLISM REVIEWS

The regulation of UDP-glucuronosyltransferase genes by tissue-specific and ligand-activated transcription factors

(2009) Peter I. Mackenzie et al.   DRUG METABOLISM REVIEWS

The prediction of drug-glucuronidation parameters in humans: UDP-glucuronosyltransferase enzyme-selective substrate and inhibitor probes for reaction phenotyping andin vitro–in vivoextrapolation of drug clearance and drug-drug interaction potential

(2009) John O. Miners et al.   DRUG METABOLISM REVIEWS

The Human UGT1A3 Enzyme Conjugates Norursodeoxycholic Acid into a C23-ester Glucuronide in the Liver

(2009) Jocelyn Trottier et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

A pharmacogenetics study of the human glucuronosyltransferase UGT1A4

(2009) Marie-Odile Benoit-Biancamano et al.   Pharmacogenetics and Genomics

Determination of mRNA Expression of Human UDP-Glucuronosyltransferases and Application for Localization in Various Human Tissues by Real-Time Reverse Transcriptase-Polymerase Chain Reaction

(2008) S. Ohno et al.   DRUG METABOLISM AND DISPOSITION