A review on cholinesterase inhibitors for Alzheimer’s disease

O-Hydroxyl- or o-amino benzylamine-tacrine hybrids: Multifunctional biometals chelators, antioxidants, and inhibitors of cholinesterase activity and amyloid-β aggregation

(2012) Fei Mao et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Inhibition of cholinesterase activity and amyloid aggregation by berberine-phenyl-benzoheterocyclic and tacrine-phenyl-benzoheterocyclic hybrids

(2012) Ling Huang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design, synthesis, and evaluation of indanone derivatives as acetylcholinesterase inhibitors and metal-chelating agents

(2012) Fan-Chao Meng et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, design and biological evaluation of novel highly potent tacrine congeners for the treatment of Alzheimer's disease

(2012) Slavka Hamulakova et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and evaluation of novel carbamate-substituted flavanone derivatives as potent acetylcholinesterase inhibitors and anti-amnestic agents

(2012) Preet Anand et al.   MEDICINAL CHEMISTRY RESEARCH

Synthesis and Biological Evaluation of Thiophene Derivatives as Acetylcholinesterase Inhibitors

(2012) Mohamed M. Ismail et al.   MOLECULES

Synthesis of New Indole Derivatives Structurally Related to Donepezil and Their Biological Evaluation as Acetylcholinesterase Inhibitors

(2012) Mohamed M. Ismail et al.   MOLECULES

Synthesis and evaluation of novel 4-[(3H,3aH,6aH)-3-phenyl)-4,6-dioxo-2-phenyldihydro-2H-pyrrolo[3,4-d]isoxazol-5(3H,6H,6aH)-yl]benzoic acid derivatives as potent acetylcholinesterase inhibitors and anti-amnestic agents

(2011) Preet Anand et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Isolation of Cholinesterase-Inhibiting Flavonoids from Morus lhou

(2011) Ji Young Kim et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Quercetin and rutin prevent scopolamine-induced memory impairment in zebrafish

(2010) S.K. Richetti et al.   BEHAVIOURAL BRAIN RESEARCH

Design, Synthesis, and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors

(2010) Leonardo Pisani et al.   ChemMedChem

Design, synthesis and evaluation of flavonoid derivatives as potent AChE inhibitors

(2009) Rong Sheng et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Tacrine-Melatonin Hybrids as Multifunctional Agents for Alzheimer's Disease, with Cholinergic, Antioxidant, and Neuroprotective Properties

(2009) María Isabel Fernández-Bachiller et al.   ChemMedChem

Structural aspects of flavonoids as inhibitors of human butyrylcholinesterase

(2009) Maja Katalinić et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Tacripyrines, the First Tacrine−Dihydropyridine Hybrids, as Multitarget-Directed Ligands for the Treatment of Alzheimer’s Disease

(2009) José Marco-Contelles et al.   JOURNAL OF MEDICINAL CHEMISTRY

New tacrine-dihydropyridine hybrids that inhibit acetylcholinesterase, calcium entry, and exhibit neuroprotection properties

(2008) Rafael León et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors

(2008) Francesco Leonetti et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design, synthesis, and acetylcholinesterase inhibitory activity of novel coumarin analogues

(2008) Xiang Zhou et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of tacrine–ferulic acid hybrids as multi-potent anti-Alzheimer drug candidates

(2008) Lei Fang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design, synthesis and evaluation of galanthamine derivatives as acetylcholinesterase inhibitors

(2008) Ping Jia et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The neuroprotective role of melatonin against amyloidβpeptide injected mice

(2008) J. Gunasingh Masilamoni et al.   FREE RADICAL RESEARCH

Synthesis and biological evaluation of novel flavonoid derivatives as dual binding acetylcholinesterase inhibitors

(2008) Yanhong Shen et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Novel Donepezil-Based Inhibitors of Acetyl- and Butyrylcholinesterase and Acetylcholinesterase-Induced β-Amyloid Aggregation

(2008) Pelayo Camps et al.   JOURNAL OF MEDICINAL CHEMISTRY

Inhibition of Acetylcholinesterase, β-Amyloid Aggregation, and NMDA Receptors in Alzheimer’s Disease: A Promising Direction for the Multi-target-Directed Ligands Gold Rush

(2008) Michela Rosini et al.   JOURNAL OF MEDICINAL CHEMISTRY

Inhibition of acetylcholinesterase by coumarins: The case of coumarin 106

(2008) A FALLARERO et al.   PHARMACOLOGICAL RESEARCH

Multi-target-directed coumarin derivatives: hAChE and BACE1 inhibitors as potential anti-Alzheimer compounds

(2007) Lorna Piazzi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS