An efficient synthesis of 3-triazolyl-2(1H)-quinolones by CuTC-catalyzed azide-alkyne cycloaddition reaction

Recent Advances in Hsp90 Inhibitors as Antitumor Agents

(2012) S. Messaoudi et al.   Anti-Cancer Agents in Medicinal Chemistry

Palladium-Catalyzed Direct Benzylation of Xanthines

(2011) Sophian Sahnoun et al.   ChemCatChem

Discovery and Biological Activity of 6BrCaQ as an Inhibitor of the Hsp90 Protein Folding Machinery

(2011) Davide Audisio et al.   ChemMedChem

Palladium-Catalyzed Coupling of 3-Halo-Substituted Coumarins, Chromenes, and Quinolones with Various Nitrogen-Containing Nucleophiles

(2011) Mohamed Ali Soussi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

1,2,3-Triazoles in Peptidomimetic Chemistry

(2011) Daniel Sejer Pedersen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Heat-shock protein 90 inhibitors as antitumor agents: a survey of the literature from 2005 to 2010

(2011) Samir Messaoudi et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

A General Copper Powder-Catalyzed Ullmann-Type Reaction of 3-Halo-4(1H)-quinolones With Various Nitrogen-Containing Nucleophiles

(2011) Davide Audisio et al.   JOURNAL OF ORGANIC CHEMISTRY

An Expeditious Copper-Catalyzed Access to 3-Aminoquinolinones, 3-Aminocoumarins and Anilines using Sodium Azide

(2010) Samir Messaoudi et al.   ADVANCED SYNTHESIS & CATALYSIS

Tricks with clicks: modification of peptidomimetic oligomers via copper-catalyzed azide-alkyne [3 + 2] cycloaddition

(2010) Justin M. Holub et al.   CHEMICAL SOCIETY REVIEWS

ATPase inhibitors of heat-shock protein 90, second season

(2010) Yves L. Janin   DRUG DISCOVERY TODAY

A Simple Synthesis of Functionalized 3-Bromocoumarins by a One-Pot Three-Component Reaction

(2010) Davide Audisio et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Pd/Cu-Catalyzed Direct Alkenylation of Azole Heterocycles with Alkenyl Halides

(2010) Sophian Sahnoun et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Transition-Metal-Catalyzed Direct C-H Alkenylation, Alkynylation, Benzylation, and Alkylation of (Hetero)arenes

(2010) Samir Messaoudi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

High Density Orthogonal Surface Immobilization via Photoactivated Copper-Free Click Chemistry

(2010) Sara V. Orski et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Site-Directed Spin-Labeling of Nucleic Acids by Click Chemistry: Detection of Abasic Sites in Duplex DNA by EPR Spectroscopy

(2010) Ulla Jakobsen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Alkyne–azide click reaction catalyzed by metallic copper under ultrasound

(2010) Pedro Cintas et al.   Nature Protocols

Monitoring Protein−Polymer Conjugation by a Fluorogenic Cu(I)-Catalyzed Azide−Alkyne 1,3-Dipolar Cycloaddition

(2009) A. (Ton) J. Dirks et al.   BIOCONJUGATE CHEMISTRY

Cu(I)-Catalyzed Huisgen Azide−Alkyne 1,3-Dipolar Cycloaddition Reaction in Nucleoside, Nucleotide, and Oligonucleotide Chemistry

(2009) Franck Amblard et al.   CHEMICAL REVIEWS

A site selective C–H arylation of free-(NH2) adenines with aryl chlorides: Application to the synthesis of 6,8-disubstituted adenines

(2009) Sophian Sahnoun et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient construction of therapeutics, bioconjugates, biomaterials and bioactive surfaces using azide–alkyne “click” chemistry☆

(2008) J LUTZ et al.   ADVANCED DRUG DELIVERY REVIEWS

Tosylcyclonovobiocic acids promote cleavage of the hsp90-associated cochaperone p23

(2008) Christine Radanyi et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Synthesis and biological activity of simplified denoviose-coumarins related to novobiocin as potent inhibitors of heat-shock protein 90 (hsp90)

(2008) Christine Radanyi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Antiproliferative and apoptotic activities of tosylcyclonovobiocic acids as potent heat shock protein 90 inhibitors in human cancer cells

(2008) Christine Radanyi et al.   CANCER LETTERS

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Microwave-assisted Pd(OH)2-catalyzed direct C−H arylation of free-(NH2) adenines with aryl halides

(2008) Sophian Sahnoun et al.   TETRAHEDRON LETTERS

Click chemistry reactions in medicinal chemistry: Applications of the 1,3-dipolar cycloaddition between azides and alkynes

(2007) Gian Cesare Tron et al.   MEDICINAL RESEARCH REVIEWS