From Anilines to Isatins: Oxidative Palladium-Catalyzed Double Carbonylation of CH Bonds

Palladium-Catalyzed Oxidative Carbonylation ofN-Allylamines for the Synthesis of β-Lactams

(2014) Wu Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct Amidation of 2′-Aminoacetophenones Using I2-TBHP: A Unimolecular Domino Approach toward Isatin and Iodoisatin

(2014) Andivelu Ilangovan et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantio- and Diastereoselective Synthesis of Spiro-epoxyoxindoles

(2014) Amina Boucherif et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-catalysed C–H activation of aliphatic amines to give strained nitrogen heterocycles

(2014) Andrew McNally et al.   NATURE

Synthesis of Isatins by I2/TBHP Mediated Oxidation of Indoles

(2014) You Zi et al.   ORGANIC LETTERS

Highly stereoselective construction of adjacent tetrasubstituted carbon stereogenic centres via an organocatalytic Mukaiyama-aldol reaction of monofluorinated silyl enol ethers to isatins

(2014) Yun-Lin Liu et al.   Organic Chemistry Frontiers

Synthesis of Dibenzopyranones through Palladium-Catalyzed Directed C-H Activation/Carbonylation of 2-Arylphenols

(2013) Shuang Luo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, synthesis and in vitro cytotoxicity evaluation of 5-(2-carboxyethenyl)isatin derivatives as anticancer agents

(2013) Kailin Han et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cu(i)-catalyzed intramolecular oxidative C–H amination of 2-aminoacetophenones: a convenient route toward isatins

(2013) Pang-Chi Huang et al.   CHEMICAL COMMUNICATIONS

Palladium-catalyzed mono- and double-carbonylation of indoles with amines controllably leading to amides and α-ketoamides

(2012) Qi Xing et al.   CHEMICAL COMMUNICATIONS

Isatins As Privileged Molecules in Design and Synthesis of Spiro-Fused Cyclic Frameworks

(2012) Girija S. Singh et al.   CHEMICAL REVIEWS

Oxidative Carbonylation as a Powerful Tool for the Direct Synthesis of Carbonylated Heterocycles

(2012) Bartolo Gabriele et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Double Carbonylation Using Near Stoichiometric Carbon Monoxide: Expedient Access to Substituted 13C2-Labeled Phenethylamines

(2012) Dennis U. Nielsen et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Oxidative Carbonylation of Benzylic C–H Bonds via Nondirected C(sp3)–H Activation

(2012) Pan Xie et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Regioselective Carbonylation of C–H Bonds of N-Alkyl Anilines for Synthesis of Isatoic Anhydrides

(2012) Zheng-Hui Guan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxidative Carbonylation Reactions: Organometallic Compounds (RM) or Hydrocarbons (RH) as Nucleophiles

(2011) Qiang Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-catalyzed carbonylative coupling reactions between Ar–X and carbon nucleophiles

(2011) Xiao-Feng Wu et al.   CHEMICAL SOCIETY REVIEWS

Synthesis ofN-Arylisatins by the Reaction of Arynes with Methyl 2-Oxo-2-(arylamino)acetates

(2011) Donald C. Rogness et al.   JOURNAL OF ORGANIC CHEMISTRY

Design of potential reverse transcriptase inhibitor containing Isatin nucleus using molecular modeling studies

(2010) Vidya Pawar et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological evaluation of 3-[4-(amino/methylsulfonyl)phenyl]methylene-indolin-2-one derivatives as novel COX-1/2 and 5-LOX inhibitors

(2010) Yisheng Lai et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2009

(2010) Roland E. Dolle et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Copper-Catalyzed Intramolecular C−H Oxidation/Acylation of Formyl-N-arylformamides Leading to Indoline-2,3-diones

(2010) Bo-Xiao Tang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd(II)-Catalyzed Carbonylation of C(sp3)−H Bonds: A New Entry to 1,4-Dicarbonyl Compounds

(2010) Eun Jeong Yoo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Room-Temperature Palladium-Catalyzed CH Activation:ortho-Carbonylation of Aniline Derivatives

(2009) Chris E. Houlden et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Carbonylation Reactions of Aryl Halides and Related Compounds

(2009) Anne Brennführer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structure-based design and parallel synthesis of N-benzyl isatin oximes as JNK3 MAP kinase inhibitors

(2009) Jingrong Cao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The alkylation of isatin-derived oximes: Spectroscopic and X-ray crystallographic structural characterization of oxime and nitrone products

(2009) Ny Sin et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Synthetic Applications of Pd(II)-Catalyzed C−H Carboxylation and Mechanistic Insights: Expedient Routes to Anthranilic Acids, Oxazolinones, and Quinazolinones

(2009) Ramesh Giri et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 1,2- and 1,3-Dicarboxylic Acids via Pd(II)-Catalyzed Carboxylation of Aryl and Vinyl C−H Bonds

(2008) Ramesh Giri et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY