A Powerful Hydrogen-Bond-Donating Organocatalyst for the Enantioselective Intramolecular Oxa-Michael Reaction of α,β-Unsaturated Amides and Esters

Streamlined Catalytic Asymmetric Synthesis of Atorvastatin

(2013) Yuji Kawato  et al.   CHEMISTRY-A EUROPEAN JOURNAL

Inner Workings of a Cinchona Alkaloid Catalyzed Oxa-Michael Cyclization: Evidence for a Concerted Hydrogen-Bond-Network Mechanism

(2013) Lukas Hintermann et al.   CHEMISTRY-A EUROPEAN JOURNAL

Structure-based ligand discovery for the Large-neutral Amino Acid Transporter 1, LAT-1

(2013) E. G. Geier et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Asymmetric Cycloetherifications by Bifunctional Aminothiourea Catalysts: The Importance of Hydrogen Bonding

(2013) Keisuke Asano et al.   SYNTHESIS-STUTTGART

Asymmetric Intramolecular Oxa-Michael Reactions of Cyclohexadienones Catalyzed by a Primary Amine Salt

(2012) Wenbin Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Enantioselective Allylic Substitution with Readily Accessible Carbonyl- and Acetal-Containing Vinylboron Reagents

(2012) Fang Gao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalyzed Isomerization of α-Substituted Alkynoates into Trisubstituted Allenoates by Dynamic Kinetic Resolution

(2012) Tsubasa Inokuma et al.   ChemCatChem

Organocatalytic asymmetric oxy-Michael addition to a γ-hydroxy-α,β-unsaturated thioester via hemiacetal intermediates

(2012) Takaaki Okamura et al.   CHEMICAL COMMUNICATIONS

DNA-based catalytic enantioselective intermolecular oxa-Michael addition reactions

(2012) Rik P. Megens et al.   CHEMICAL COMMUNICATIONS

Efficient copper-catalyzed Michael addition of acrylic derivatives with primary alcohols in the presence of base

(2012) Feng Wang et al.   CHEMICAL COMMUNICATIONS

Asymmetric Ion-Pairing Catalysis of the Reversible Cyclization of 2′-Hydroxychalcone to Flavanone: Asymmetric Catalysis of an Equilibrating Reaction

(2012) Lukas Hintermann et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

An Asymmetric Synthesis of 1,2,4-Trioxane Anticancer Agents via Desymmetrization of Peroxyquinols through a Brønsted Acid Catalysis Cascade

(2012) David M. Rubush et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective formal hydration of α,β-unsaturated acceptors: asymmetric conjugate addition of silicon and boron nucleophiles

(2011) Eduard Hartmann et al.   CHEMICAL COMMUNICATIONS

Recent developments in the field of oxa-Michael reactions

(2011) Carl F. Nising et al.   CHEMICAL SOCIETY REVIEWS

Bifunctional Hydrogen-Bond Donors That Bear a Quinazoline or Benzothiadiazine Skeleton for Asymmetric Organocatalysis

(2011) Tsubasa Inokuma et al.   CHEMISTRY-A EUROPEAN JOURNAL

Chiba-G-Catalyzed Intramolecular Oxo-Michael Addition: Synthetic Approaches to Vitamin E Skeleton

(2011) Tsutomu Ishikawa et al.   HETEROCYCLES

The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates

(2011) Stephen D. Roughley et al.   JOURNAL OF MEDICINAL CHEMISTRY

Stereoselective Synthesis of 2,6-Cis-Substituted Tetrahydropyrans: Brønsted Acid-Catalyzed Intramolecular Oxa-Conjugate Cyclization of α,β-Unsaturated Ester Surrogates

(2011) Haruhiko Fuwa et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Catalytic Cycloetherification Mediated by Bifunctional Organocatalysts

(2011) Keisuke Asano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Organocascade Kinetic Resolution

(2011) Patrick G. McGarraugh et al.   ORGANIC LETTERS

Development of Chiral Thiourea Catalysts and Its Application to Asymmetric Catalytic Reactions

(2010) Yoshiji Takemoto   CHEMICAL & PHARMACEUTICAL BULLETIN

Synthesis of 2-Isoxazolines: Enantioselective and Racemic Methods Based on Conjugate Additions of Oximes

(2010) Antti Pohjakallio et al.   CHEMISTRY-A EUROPEAN JOURNAL

Desymmetrization of Cyclohexadienones via Brønsted Acid-Catalyzed Enantioselective Oxo-Michael Reaction

(2010) Qing Gu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic enantioselective syn hydration of enones in water using a DNA-based catalyst

(2010) Arnold J. Boersma et al.   Nature Chemistry

Asymmetric organocatalytic synthesis of six-membered oxygenated heterocycles

(2010) Marta G. Núñez et al.   TETRAHEDRON

A novel one-step method for the reductive allylation of esters and the first total synthesis of (±)-erythrococcamide B

(2010) Roman Lagoutte et al.   TETRAHEDRON LETTERS

Novel Cinchona-Aminobenzimidazole Bifunctional Organocatalysts

(2009) Lei Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Organocatalytic Domino Oxa-Michael/Aldol/Hemiacetalization: Synthesis of Polysubstituted Furofuranes Containing Four Stereocenters

(2009) Efraím Reyes et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Redox Economy in Organic Synthesis

(2009) Noah Z. Burns et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral 2-Aminobenzimidazoles as Recoverable Organocatalysts for the Addition of 1,3-Dicarbonyl Compounds to Nitroalkenes†

(2009) Diana Almaşi et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Asymmetric Formal [3 + 2] Cycloaddition with in Situ-GeneratedN-Carbamoyl Nitrones

(2009) Claudio Gioia et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hydroxyl Group-Directed Organocatalytic Asymmetric Michael Addition of α,β-Unsaturated Ketones with Alkenylboronic Acids

(2009) Tsubasa Inokuma et al.   ORGANIC LETTERS

Organocatalytic Synthesis of an Alkyltetrahydropyran

(2009) D. Díez et al.   SYNLETT

The oxa-Michael reaction: from recent developments to applications in natural product synthesis

(2008) Carl F. Nising et al.   CHEMICAL SOCIETY REVIEWS

Guanidine-Catalyzed Asymmetric Synthesis of 2,2-Disubstituted Chromane Skeletons by Intramolecular Oxa-Michael Addition

(2008) Noriko Saito et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Epi-Cinchona Based Thiourea Organocatalyst Family as an Efficient Asymmetric Michael Addition Promoter: Enantioselective Conjugate Addition of Nitroalkanes to Chalcones and α,β-UnsaturatedN-Acylpyrroles

(2008) Benedek Vakulya et al.   JOURNAL OF ORGANIC CHEMISTRY

Chiral Squaramide Derivatives are Excellent Hydrogen Bond Donor Catalysts

(2008) Jeremiah P. Malerich et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective, Organocatalytic Oxy-Michael Addition to γ/δ-Hydroxy-α,β-enones:  Boronate-Amine Complexes as Chiral Hydroxide Synthons

(2007) De Run Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY