Dynamic Combinatorial Chemistry Employing Boronic Acids/Boronate Esters Leads to Potent Oxygenase Inhibitors

Inhibition of 2-oxoglutarate dependent oxygenases

(2011) Nathan R. Rose et al.   CHEMICAL SOCIETY REVIEWS

An approach to enzyme inhibition employing reversible boronate ester formation

(2011) Ivanhoe K. H. Leung et al.   MedChemComm

Selective Inhibitors of the JMJD2 Histone Demethylases: Combined Nondenaturing Mass Spectrometric Screening and Crystallographic Approaches

(2010) Nathan R. Rose et al.   JOURNAL OF MEDICINAL CHEMISTRY

Using NMR Solvent Water Relaxation to Investigate Metalloenzyme−Ligand Binding Interactions

(2009) Ivanhoe K. H. Leung et al.   JOURNAL OF MEDICINAL CHEMISTRY

Structural Basis for Binding of Hypoxia-Inducible Factor to the Oxygen-Sensing Prolyl Hydroxylases

(2009) Rasheduzzaman Chowdhury et al.   STRUCTURE

Water-Based Ligand Screening for Paramagnetic Metalloproteins

(2008) Ivano Bertini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dynamic Combinatorial Mass Spectrometry Leads to Metallo-β-lactamase Inhibitors

(2008) Benoît M. R. Liénard et al.   JOURNAL OF MEDICINAL CHEMISTRY