“Triazole Bridge”: Disulfide-Bond Replacement by Ruthenium-Catalyzed Formation of 1,5-Disubstituted 1,2,3-Triazoles

Implication of the disulfide bridge in trypsin inhibitor SFTI-1 in its interaction with serine proteinases

(2010) Anna Łęgowska et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Oxidative folding of hepcidin at acidic pH

(2010) Jingwen Zhang et al.   BIOPOLYMERS

Development of a Functional cis-Prolyl Bond Biomimetic and Mechanistic Implications for Nickel Superoxide Dismutase

(2010) Daniel Tietze et al.   CHEMISTRY-A EUROPEAN JOURNAL

Optimization of oxidative folding methods for cysteine-rich peptides: a study of conotoxins containing three disulfide bridges

(2010) Andrew M. Steiner et al.   JOURNAL OF PEPTIDE SCIENCE

Solving the α-Conotoxin Folding Problem: Efficient Selenium-Directed On-Resin Generation of More Potent and Stable Nicotinic Acetylcholine Receptor Antagonists

(2010) Markus Muttenthaler et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

“Clicktophycin-52”: A Bioactive Cryptophycin-52 Triazole Analogue

(2010) Markus Nahrwold et al.   ORGANIC LETTERS

Analogues of Trypsin Inhibitor SFTI-1 with Disulfide Bridge Substituted by Various Length of Carbonyl Bridges

(2010) Anna Legowska et al.   PROTEIN AND PEPTIDE LETTERS

Conformationally Homogeneous Heterocyclic Pseudotetrapeptides as Three-Dimensional Scaffolds for Rational Drug Design: Receptor-Selective Somatostatin Analogues

(2009) John M. Beierle et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Probing the Bioactive Conformation of an Archetypal Natural Product HDAC Inhibitor with Conformationally Homogeneous Triazole-Modified Cyclic Tetrapeptides

(2009) W. Seth Horne et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Establishing regiocontrol of disulfide bond isomers of α-conotoxin ImI via the synthesis of N-to-C cyclic analogs

(2009) Christopher J. Armishaw et al.   BIOPOLYMERS

Cyclotides: macrocyclic peptides with applications in drug design and agriculture

(2009) David J. Craik et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

Biological diversity and therapeutic potential of natural and engineered cystine knot miniproteins

(2009) Harald Kolmar   CURRENT OPINION IN PHARMACOLOGY

Peptide Cyclization and Cyclodimerization by CuI-Mediated Azide−Alkyne Cycloaddition

(2009) Reshma Jagasia et al.   JOURNAL OF ORGANIC CHEMISTRY

Side chain-to-side chain cyclization by click reaction

(2009) Alexandra Le Chevalier Isaad et al.   JOURNAL OF PEPTIDE SCIENCE

Sunflower Trypsin Inhibitor 1 Derivatives as Molecular Scaffolds for the Development of Novel Peptidic Radiopharmaceuticals

(2009) Regine García Boy et al.   MOLECULAR IMAGING AND BIOLOGY

Electronic Structure of the Azide Group in 3¢-Azido-3¢-deoxythymidine (AZT) Compared to Small Azide Compounds

(2009) Fang-Fang Chen et al.   MOLECULES

Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity

(2009) Mohammed Akhter Hossain et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Application of copper(i) catalyzed azide–alkyne [3+2] cycloaddition to the synthesis of template-assembled multivalent peptide conjugates

(2009) Olga Avrutina et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Accessing Skeletal Diversity Using Catalyst Control: Formation ofnandn+ 1 Macrocyclic Triazole Rings

(2009) Ann Rowley Kelly et al.   ORGANIC LETTERS

Efficient construction of therapeutics, bioconjugates, biomaterials and bioactive surfaces using azide–alkyne “click” chemistry☆

(2008) J LUTZ et al.   ADVANCED DRUG DELIVERY REVIEWS

Structurally Minimized μ-Conotoxin Analogues as Sodium Channel Blockers: Implications for Designing Conopeptide-Based Therapeutics

(2008) Tiffany S. Han et al.   ChemMedChem

Synthesis and Conformational Analysis of a Cyclic Peptide Obtained viaitoi+4 Intramolecular Side-Chain to Side-Chain Azide−Alkyne 1,3-Dipolar Cycloaddition

(2008) Sonia Cantel et al.   JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Click chemistry reactions in medicinal chemistry: Applications of the 1,3-dipolar cycloaddition between azides and alkynes

(2007) Gian Cesare Tron et al.   MEDICINAL RESEARCH REVIEWS