The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist

Ghrelin receptor antagonism attenuates nicotine-induced locomotor stimulation, accumbal dopamine release and conditioned place preference in mice

(2011) Elisabet Jerlhag et al.   DRUG AND ALCOHOL DEPENDENCE

Ghrelin directly targets the ventral tegmental area to increase food motivation

(2011) K.P. Skibicka et al.   NEUROSCIENCE

The Ghrelin Signalling System Is Involved in the Consumption of Sweets

(2011) Sara Landgren et al.   PLoS One

Pharmacologic antagonism of ghrelin receptors attenuates development of nicotine induced locomotor sensitization in rats

(2011) Paul J. Wellman et al.   REGULATORY PEPTIDES

Ghrelin increases intake of rewarding food in rodents

(2010) Emil Egecioglu et al.   ADDICTION BIOLOGY

Ghrelin Receptor Antagonism Decreases Alcohol Consumption and Activation of Perioculomotor Urocortin-Containing Neurons

(2010) Simranjit Kaur et al.   ALCOHOLISM-CLINICAL AND EXPERIMENTAL RESEARCH

Acute and chronic suppression of the central ghrelin signaling system reveals a role in food anticipatory activity

(2010) Linda A.W. Verhagen et al.   EUROPEAN NEUROPSYCHOPHARMACOLOGY

Ghrelin receptor antagonism attenuates cocaine- and amphetamine-induced locomotor stimulation, accumbal dopamine release, and conditioned place preference

(2010) Elisabet Jerlhag et al.   PSYCHOPHARMACOLOGY

Anorexigenic and electrophysiological actions of novel ghrelin receptor (GHS-R1A) antagonists in rats

(2009) Nicolas Salomé et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

On the Central Mechanism Underlying Ghrelin’s Chronic Pro-Obesity Effects in Rats: New Insights from Studies Exploiting a Potent Ghrelin Receptor Antagonist

(2009) N. Salomé et al.   JOURNAL OF NEUROENDOCRINOLOGY

Reduced anticipatory locomotor responses to scheduled meals in ghrelin receptor deficient mice

(2009) I.D. Blum et al.   NEUROSCIENCE

Requirement of central ghrelin signaling for alcohol reward

(2009) E. Jerlhag et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Stomach ghrelin-secreting cells as food-entrainable circadian clocks

(2009) J. LeSauter et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Whole body and tissue imaging of the butyrylcholinesterase knockout mouse injected with near infrared dye labeled butyrylcholinesterase

(2008) Ellen G. Duysen et al.   CHEMICO-BIOLOGICAL INTERACTIONS

New Trisubstituted 1,2,4-Triazole Derivatives as Potent Ghrelin Receptor Antagonists. 3. Synthesis and Pharmacological in Vitro and in Vivo Evaluations

(2008) Aline Moulin et al.   JOURNAL OF MEDICINAL CHEMISTRY

Trisubstituted 1,2,4-triazoles as ligands for the ghrelin receptor: On the significance of the orientation and substitution at position 3

(2007) Aline Moulin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS