Regioselective and Stereoselective [3+3] Annulation of Ketones Derived Azomethine Ylides with 2-Indolylethylenes: Direct Access to Highly Substituted Tetrahydro-γ-Carbolines

[3 + 3] Cycloaddition of in Situ Formed Azaoxyallyl Cations with 2-Alkenylindoles: An Approach to Tetrahydro-β-carbolinones

(2017) Kaifan Zhang et al.   ORGANIC LETTERS

Recent advances in the enantioselective 1,3-dipolar cycloaddition of azomethine ylides and dipolarophiles

(2017) Bilel Bdiri et al.   TETRAHEDRON-ASYMMETRY

Cu(i)-catalyzed Michael addition of ketiminoesters to β-trifluoromethyl β,β-disubstituted enones: rapid access to 1-pyrrolines bearing a quaternary all-carbon stereocenter

(2017) Bing Liu et al.   Organic Chemistry Frontiers

Catalytic Enantioselective and Regioselective [3+3] Cycloadditions Using 2-Indolylmethanols as 3 C Building Blocks

(2016) Xiao-Xue Sun et al.   CHEMISTRY-A EUROPEAN JOURNAL

Cu(I)-Catalyzed Chemoselective and Stereoselective [3 + 3] Cycloaddition of Azomethine Ylides with 2-Indolylnitroethylenes: Facile Access to Highly Substituted Tetrahydro-γ-Carbolines

(2016) Wu-Lin Yang et al.   ACS Catalysis

Recent Advances of Catalytic Asymmetric 1,3-Dipolar Cycloadditions

(2015) Takuya Hashimoto et al.   CHEMICAL REVIEWS

Ervatamines A–I, Anti-inflammatory Monoterpenoid Indole Alkaloids with Diverse Skeletons from Ervatamia hainanensis

(2015) Dong-Bo Zhang et al.   JOURNAL OF NATURAL PRODUCTS

Enantiodivergent Synthesis of Bis-Spiropyrrolidines via Sequential Interrupted and Completed (3 + 2) Cycloadditions

(2015) Egoitz Conde et al.   JOURNAL OF ORGANIC CHEMISTRY

Construction of Benzo[c]carbazoles and Their Antitumor Derivatives through the Diels–Alder Reaction of 2-Alkenylindoles and Arynes

(2015) Feng Sha et al.   JOURNAL OF ORGANIC CHEMISTRY

Exoselective 1,3-Dipolar [3 + 6] Cycloaddition of Azomethine Ylides with 2-Acylcycloheptatrienes: Stereoselectivity and Mechanistic Insight

(2015) Zhao-Lin He et al.   ORGANIC LETTERS

Brucine Diol–Copper-Catalyzed Asymmetric Synthesis of endo-Pyrrolidines: The Mechanistic Dichotomy of Imino Esters

(2015) Jian-Yuan Li et al.   ORGANIC LETTERS

Silver-catalyzed asymmetric Michael addition of azomethine ylide to arylidene diphosphonates using ThioClickFerrophos ligand

(2015) Midori Kimura et al.   TETRAHEDRON LETTERS

Direct Asymmetric Synthesis of β-Bis-Aryl-α-Amino Acid Esters via Enantioselective Copper-Catalyzed Addition of p-Quinone Methides

(2015) Fu-Sheng He et al.   ACS Catalysis

Chiral Fullerenes from Asymmetric Catalysis

(2014) Enrique E. Maroto et al.   ACCOUNTS OF CHEMICAL RESEARCH

Catalytic Enantioselective 1,3-Dipolar Cycloadditions of Azomethine Ylides for Biology-Oriented Synthesis

(2014) Rishikesh Narayan et al.   ACCOUNTS OF CHEMICAL RESEARCH

Catalytic Asymmetric Formal [3+3] Cycloaddition of an Azomethine Ylide with 3-Indolylmethanol: Enantioselective Construction of a Six-Membered Piperidine Framework

(2014) Feng Shi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Diastereo- and Enantioselective Construction of a Bispirooxindole Scaffold Containing a Tetrahydro-β-carboline Moiety through an Organocatalytic Asymmetric Cascade Reaction

(2014) Wei Dai et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric 1,3-Dipolar [3 + 6] Cycloaddition of Azomethine Ylides with 2-Acyl Cycloheptatrienes: Efficient Construction of Bridged Heterocycles Bearing Piperidine Moiety

(2014) Qing-Hua Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(I)-Catalyzed Regio- and Stereoselective [6 + 3] Cycloaddition of Azomethine Ylides with Tropone: An Efficient Asymmetric Access to Bridged Azabicyclo[4.3.1]decadienes

(2014) Huai-Long Teng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Catalyzed [6 + 3] Cycloaddition of Tropone with Azomethine Ylides: A Practical Access to Piperidine-Fused Bicyclic Heterocycles

(2014) Honglei Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(I)-Catalyzed Highly Enantioselective [3 + 3] Cycloaddition between Two Different 1,3-Dipoles, Phthalazinium Dicyanomethanides and Iminoester-Derived Azomethine Ylides

(2014) Chunhao Yuan et al.   ORGANIC LETTERS

Novel Carboline Derivatives as Potent Antifungal Lead Compounds: Design, Synthesis, and Biological Evaluation

(2014) Shengzheng Wang et al.   ACS Medicinal Chemistry Letters

Chiral Brønsted Acid Catalyzed Stereoselective [3+3] Cycloaddition Reaction of Azomethine Ylide to Vinylimine Intermediates: Constructing Fully Functionalized Chiral Tetrahydro-β-Carboline

(2013) Jianzhou Huang et al.   ACTA CHIMICA SINICA

Synthesis of Glutamic Acid and Highly Functionalized Pyrrolidine Derivatives by Utilizing Tunable Calcium Catalysts for Chemoselective Asymmetric 1,4-Addition and [3+2] Cycloaddition Reactions

(2013) Martin Hut'ka et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Copper-Catalyzed [3+3] Cycloaddition of Azomethine Ylides with Azomethine Imines

(2013) Hongchao Guo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fulvenes as Effective Dipolarophiles in Copper(I)-Catalyzed [6+3] Cycloaddition of Azomethine Ylides: Asymmetric Construction of Piperidine Derivatives

(2013) Zhao-Lin He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric 1,3-Dipolar Cycloaddition of Two Different Ylides: Facile Access to Chiral 1,2,4-Triazinane Frameworks

(2013) Min-Chao Tong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Identification of 2-(2-(1-Naphthoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5(2H)-yl)acetic Acid (Setipiprant/ACT-129968), a Potent, Selective, and Orally Bioavailable Chemoattractant Receptor-Homologous Molecule Expressed on Th2 Cells (CRTH2) Antagonist

(2013) Heinz Fretz et al.   JOURNAL OF MEDICINAL CHEMISTRY

Silver/ThioClickFerrophos Complex as an Effective Catalyst for Asymmetric Conjugate Addition of Glycine Imino Ester to Unsaturated Malonates and α-Enones

(2013) Takashi Konno et al.   ORGANIC LETTERS

Highly Enantioselective Catalytic [6+3] Cycloadditions of Azomethine Ylides

(2012) Marco Potowski et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Silver/ThioClickFerrophos-Catalyzed Enantioselective Conjugate Addition and Cycloaddition of Glycine Imino Ester with Nitroalkenes

(2012) Kazumi Imae et al.   ORGANIC LETTERS

Novel dipolarophiles and dipoles in the metal-catalyzed enantioselective 1,3-dipolar cycloaddition of azomethine ylides

(2011) Javier Adrio et al.   CHEMICAL COMMUNICATIONS

Enantiocontrolled Synthesis of β-Branched α-Amino Acids by Using CuI-Catalyzed 1,4-Addition of Glycine Imines to β-Substituted gem-Diactivated Olefins

(2011) Jorge Hernández-Toribio et al.   CHEMISTRY-A EUROPEAN JOURNAL

Stereodivergency in Catalytic Asymmetric Conjugate Addition Reactions of Glycine (Ket)imines

(2011) Hun Young Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Ferrocenyl-DHIPOH/Cu(OAc)2Complex for Diastereo- and Enantioselective Catalysis of the 1,4-Addition of Glycine Derivatives to Alkylidene Malonates

(2011) Yu-Hua Shi et al.   ORGANIC LETTERS

Novel N,O-Cu(OAc)2 complex catalysed diastereo- and enantioselective 1,4-addition of glycine derivatives to alkylidene malonates

(2011) Ming Wang et al.   Catalysis Science & Technology

Synthesis and biological activity of N-aroyl-tetrahydro-γ-carbolines

(2010) Alexandre Bridoux et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Cu-Catalyzed Asymmetric Michael Addition of Glycine Derivatives to α,β-Unsaturated Malonates

(2010) Xuelong Hou et al.   CHINESE JOURNAL OF CHEMISTRY

Diastereo- and Enantioselective Synthesis of α,γ-Diaminobutyric Acid Derivatives via Cu-Catalyzed Asymmetric Michael Reaction

(2010) Qing Li et al.   ORGANIC LETTERS

Synthesis and biological activity of 5-styryl and 5-phenethyl-substituted 2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indoles

(2009) Alexandre V. Ivachtchenko et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Substrate-Controlled Diastereoselectivity Switch in Catalytic Asymmetric Direct Mannich Reaction of Glycine Derivatives with Imines: Fromanti- tosyn-α,β-Diamino Acids

(2009) Jorge Hernández-Toribio et al.   CHEMISTRY-A EUROPEAN JOURNAL

Two Indolotryptanthrin Alkaloids from Cephalantheropsis gracilis

(2009) Pei-Lin Wu et al.   HETEROCYCLES

Highly Enantioselective Cu-Catalyzed Conjugate Addition−Elimination of Activated Allylic Acetates with Glycine Derivatives

(2009) Chun-Gen Chen et al.   ORGANIC LETTERS

Development of Catalytic Asymmetric 1,4-Addition and [3 + 2] Cycloaddition Reactions Using Chiral Calcium Complexes

(2008) Tetsu Tsubogo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Calcium-Catalyzed Diastereo- and Enantioselective 1,4-Addition of Glycine Derivatives to α,β-Unsaturated Esters

(2008) Shū Kobayashi et al.   ORGANIC LETTERS