Copper-Catalyzed Intermolecular Oxidative Cyclization of Halo- alkynes: Synthesis of 2-Halo-substituted Imidazo[1,2-a]pyridines, Imidazo[1,2-a]pyrazines and Imidazo[1,2-a]pyrimidines

Catalytic Electrophilic Halogenation of Silyl-Protected and Terminal Alkynes: Trapping Gold(I) Acetylidesvs. a Brønsted Acid-Promoted Reaction

(2012) Pavel Starkov et al.   ADVANCED SYNTHESIS & CATALYSIS

Silver-Assisted Difunctionalization of Terminal Alkynes: Highly Regio- and Stereoselective Synthesis of Bromofluoroalkenes

(2012) Yibiao Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium(II)-Catalyzed Intramolecular Diamination of Alkynes under Aerobic Oxidative Conditions: Catalytic Turnover of an Iodide Ion

(2012) Bo Yao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Heteroaromatic imidazo[1,2-a]pyridines synthesis from C–H/N–H oxidative cross-coupling/cyclization

(2012) Chuan He et al.   CHEMICAL COMMUNICATIONS

Cu(I)-Catalyzed Synthesis of Imidazo[1,2-a]pyridines from Aminopyridines and Nitroolefins Using Air as the Oxidant

(2012) Ru-Long Yan et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal Cocatalyzed Tandem Alkynylative Cyclization Reaction of in Situ Formed N-Iminoisoquinolinium Ylides with Bromoalkynes via C–H Bond Activation

(2012) Ping Huang et al.   JOURNAL OF ORGANIC CHEMISTRY

Imidazo[1,2-a]pyridines Susceptible to Excited State Intramolecular Proton Transfer: One-Pot Synthesis via an Ortoleva–King Reaction

(2012) Anton J. Stasyuk et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Aerobic [3+2]-Annulation of N-Alkenyl Amidines

(2012) Yi-Feng Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(II)-Catalyzed Synthesis of Naphthalene-1,3-diamine Derivatives from Haloalkynes and Amines

(2012) Zhengwang Chen et al.   ORGANIC LETTERS

Intramolecular Oxidative Diamination and Aminohydroxylation of Olefins under Metal-Free Conditions

(2012) Hyun Jin Kim et al.   ORGANIC LETTERS

Copper(II)/Iron(III) Co-catalyzed Intermolecular Diamination of Alkynes: Facile Synthesis of Imidazopyridines

(2012) Jing Zeng et al.   ORGANIC LETTERS

Copper-Catalyzed Intramolecular Dehydrogenative Aminooxygenation: Direct Access to Formyl-Substituted Aromatic N-Heterocycles

(2011) Honggen Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

TBAI-catalyzed oxidative coupling of aminopyridines with β-keto esters and 1,3-diones—synthesis of imidazo[1,2-a]pyridines

(2011) Lijuan Ma et al.   CHEMICAL COMMUNICATIONS

Systematic Structure Modifications of Imidazo[1,2-a]pyrimidine to Reduce Metabolism Mediated by Aldehyde Oxidase (AO)

(2011) Angelica Linton et al.   JOURNAL OF MEDICINAL CHEMISTRY

Enantioselective Alkynylation of Aldehydes with 1-Haloalkynes Catalyzed by Tethered Bis(8-quinolinato) Chromium Complex

(2011) Dmitry L. Usanov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Direct Ethynylation of C(sp3)–H Bonds in Aliphatic Carboxylic Acid Derivatives

(2011) Yusuke Ano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct preparation of thiazoles, imidazoles, imidazopyridines and thiazolidines from alkenes

(2011) Timothy J. Donohoe et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Introducing a New Class ofN-Phosphoryl Ynamides via Cu(I)-Catalyzed Amidations of Alkynyl Bromides

(2011) Kyle A. DeKorver et al.   ORGANIC LETTERS

Sequential and One-Pot Reactions of Phenols with Bromoalkynes for the Synthesis of (Z)-2-Bromovinyl Phenyl Ethers and Benzo[b]furans

(2011) Shihua Wang et al.   ORGANIC LETTERS

Copper-Catalyzed Synthesis of Quinoxalines witho-Phenylenediamine and Terminal Alkyne in the Presence of Bases

(2011) Wen Wang et al.   ORGANIC LETTERS

Cationic Gold Catalyzes ω-Bromination of Terminal Alkynes and Subsequent Hydroaddition Reactions

(2011) Antonio Leyva-Pérez et al.   ACS Catalysis

An Intermolecular Palladium-Catalyzed Diamination of Unactivated Alkenes

(2010) Álvaro Iglesias et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Formal Inverse Sonogashira Reaction: Direct Alkynylation of Arenes and Heterocycles with Alkynyl Halides

(2010) Alexander S. Dudnik et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Promoted and Copper-Catalyzed Intermolecular Alkene Diamination

(2010) Fatima C. Sequeira et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

General and Efficient Copper-Catalyzed Three-Component Coupling Reaction towards Imidazoheterocycles: One-Pot Synthesis of Alpidem and Zolpidem

(2010) Natalia Chernyak et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The use of Br/Cl to promote regioselective gold-catalyzed rearrangement of propargylic carboxylates: an efficient synthesis of (1Z, 3E)-1-bromo/chloro-2-carboxy-1,3-dienes

(2010) Yanzhao Wang et al.   CHEMICAL COMMUNICATIONS

A Direct Intramolecular C−H Amination Reaction Cocatalyzed by Copper(II) and Iron(III) as Part of an Efficient Route for the Synthesis of Pyrido[1,2-a]benzimidazoles fromN-Aryl-2-aminopyridines

(2010) Honggen Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthetic and Mechanistic Studies on Pd(0)-Catalyzed Diamination of Conjugated Dienes

(2010) Baoguo Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(I)−Amido Complexes in the Ullmann Reaction: Reactions of Cu(I)−Amido Complexes with Iodoarenes with and without Autocatalysis by CuI

(2010) Ramesh Giri et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(I)-Catalyzed Regioselective Diamination of Conjugated Dienes via Dual Mechanistic Pathways

(2010) Baoguo Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Aerobic Oxidative Functionalization of an Arene C−H Bond: Evidence for an Aryl-Copper(III) Intermediate

(2010) Amanda E. King et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Silver-Catalyzed Difunctionalization of Terminal Alkynes: Highly Regio- and Stereoselective Synthesis of (Z)-β-Haloenol Acetates

(2010) Zhengwang Chen et al.   ORGANIC LETTERS

Copper-Catalyzed Synthesis of N-Fused Heterocycles through Regioselective 1,2-Aminothiolation of 1,1-Dibromoalkenes

(2010) Hui Xu et al.   ORGANIC LETTERS

Complementary Regioselectivity in the Cu(I)-Catalyzed Diamination of Conjugated Dienes To Form Cyclic Sulfamides

(2010) Richard G. Cornwall et al.   ORGANIC LETTERS

Direct Preparation of Heteroaromatic Compounds from Alkenes

(2010) Timothy Donohoe et al.   SYNLETT

Direct observation of CuI/CuIII redox steps relevant to Ullmann-type coupling reactions

(2010) Alicia Casitas et al.   Chemical Science

Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes

(2009) Jason E. Hein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper as a Powerful Catalyst in the Direct Alkynylation of Azoles

(2009) François Besselièvre et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

3-(3-Aryloxyaryl)imidazo[1,2-a]pyridine sulfones as liver X receptor agonists

(2009) Robert R. Singhaus et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Scaffold hopping from pyridones to imidazo[1,2-a]pyridines. New positive allosteric modulators of metabotropic glutamate 2 receptor

(2009) Gary Tresadern et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Mechanism ofN-Fluorobenzenesulfonimide Promoted Diamination and Carboamination Reactions: Divergent Reactivity of a Pd(IV) Species

(2009) Paul A. Sibbald et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Antidepressants for the Treatment of Insomnia

(2008) Michael H Wiegand   DRUGS

2-Phenyl-imidazo[1,2-a]pyridine Compounds Containing Hydrophilic Groups as Potent and Selective Ligands for Peripheral Benzodiazepine Receptors: Synthesis, Binding Affinity and Electrophysiological Studies

(2008) Nunzio Denora et al.   JOURNAL OF MEDICINAL CHEMISTRY

Structural Requirements for Eszopiclone and Zolpidem Binding to the γ-Aminobutyric Acid Type-A (GABAA) Receptor Are Different

(2008) Susan M. Hanson et al.   JOURNAL OF MEDICINAL CHEMISTRY

Energies of Low-Lying Excited States of Linear Polyenes

(2008) Ronald L. Christensen et al.   JOURNAL OF PHYSICAL CHEMISTRY A

Dual Role of Alkynyl Halides in One-Step Synthesis of Alkynyl Epoxides

(2008) Alexander Trofimov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed 1,2-Double Amination of 1-Halo-1-alkynes. Concise Synthesis of Protected Tetrahydropyrazines and Related Heterocyclic Compounds

(2008) Yasuhiro Fukudome et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper Catalyzed Enantioselective Intramolecular Aminooxygenation of Alkenes

(2008) Peter H. Fuller et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY