Journal
ADVANCED SYNTHESIS & CATALYSIS
Volume 355, Issue 4, Pages 711-715Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/adsc.201200997
Keywords
arylhydrazines; 3-aryl-1H-indoles; CH activation; denitrogenative process; palladium-catalyzed reaction
Categories
Funding
- National Science Foundation of P. R. China [J1103307]
Ask authors/readers for more resources
A novel palladium-catalyzed approach to direct C-3-arylation of 1H-indoles with arylhydrazines using air as the oxidant via CN bond cleavage has been developed. Various substituents are tolerated in this system in moderate to good yields. This reaction could also be compatible with a larger scale. Thus, this strategy using arylhydrazines as arylating reagents provides a powerful method for constructing substituted 3-aryl-1H-indoles.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available