Base-Mediated Direct Arylation of Pyrrole Derivatives

Regioselective Functionalization of the Imidazole Ring via Transition Metal-Catalyzed CN and CC Bond Forming Reactions

(2010) Fabio Bellina et al.   ADVANCED SYNTHESIS & CATALYSIS

Retraction: Facile Palladium-Catalyzed Arylation of Heterocycles and Nonactivated Arenes with Aryl Chlorides

(2010) Jan Pschierer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-Catalyzed Direct Arylation of Unactivated Arenes with Aryl Halides

(2010) Wei Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed Direct CH Arylation and Alkenylation of Heteroarenes with Organosilicon Reagents

(2010) Hitoshi Hachiya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Triethanolamine-Mediated Palladium-Catalyzed Regioselective C-2 Direct Arylation of Free NH-Pyrroles

(2010) Farnaz Jafarpour et al.   JOURNAL OF ORGANIC CHEMISTRY

C−H Bonds as Ubiquitous Functionality: A General Approach to Complex Arylated Imidazoles via Regioselective Sequential Arylation of All Three C−H Bonds and RegioselectiveN-Alkylation Enabled by SEM-Group Transposition

(2010) Jung Min Joo et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalysis in Cross-Coupling: DMEDA-Catalyzed Direct C−H Arylation of Unactivated Benzene

(2010) Wei Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An efficient organocatalytic method for constructing biaryls through aromatic C–H activation

(2010) Chang-Liang Sun et al.   Nature Chemistry

When is free really free?

(2010) Nicholas E. Leadbeater   Nature Chemistry

Metal-Free Coupling of Azoles with 2- and 3-Haloindoles Providing Access to Novel 2- or 3-(Azol-1-yl)indole Derivatives

(2010) Martin Poirier et al.   ORGANIC LETTERS

Room-Temperature Direct Arylation of Polyfluorinated Arenes under Biphasic Conditions

(2010) Olivier René et al.   ORGANIC LETTERS

Iron-Mediated Direct Suzuki−Miyaura Reaction: A New Method for theortho-Arylation of Pyrrole and Pyridine

(2010) Jun Wen et al.   ORGANIC LETTERS

Efficient Cross-Coupling Reactions of Nitrogen Nucleophiles with Aryl Halides in Water

(2009) Yong-Chua Teo   ADVANCED SYNTHESIS & CATALYSIS

Transition Metal-Catalysed, Direct and Site-Selective N1-, C2- or C3-Arylation of the Indole Nucleus: 20 Years of Improvements

(2009) Lionel Joucla et al.   ADVANCED SYNTHESIS & CATALYSIS

Iron-Catalyzed Chemoselective ortho Arylation of Aryl Imines by Directed CH Bond Activation

(2009) Naohiko Yoshikai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Direct C Arylation of Heterocycles with Aryl Bromides: Discovery of Fluorescent Core Frameworks

(2009) Dongbing Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

On the Role of Metal Contaminants in Catalyses with FeCl3

(2009) Stephen L. Buchwald et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(II)-Catalyzed CH Activation/CC Cross-Coupling Reactions: Versatility and Practicality

(2009) Xiao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Aluminum Bases for the Highly Chemoselective Preparation of Aryl and Heteroaryl Aluminum Compounds

(2009) Stefan H. Wunderlich et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed C3 or C4 Direct Arylation of Heteroaromatic Compounds with Aryl Halides by CH Bond Activation

(2009) Julien Roger et al.   ChemCatChem

Copper-catalyzed arene C–H bond cross-coupling

(2009) Hien-Quang Do et al.   CHEMICAL COMMUNICATIONS

Palladium-Catalysed Direct 3- or 4-Arylation of 2,5-Disubstituted Pyrrole Derivatives: An Economically and Environmentally Attractive Procedure

(2009) Yacoub Fall et al.   ChemSusChem

Synthesis of 3-Aryl-8-oxo-5,6,7,8-tetrahydroindolizines via a Palladium-Catalyzed Arylation and Heteroarylation

(2009) Stéphanie Gracia et al.   JOURNAL OF ORGANIC CHEMISTRY

Establishment of Broadly Applicable Reaction Conditions for the Palladium-Catalyzed Direct Arylation of Heteroatom-Containing Aromatic Compounds

(2009) Benoît Liégault et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed 2-Arylation of Pyrroles

(2009) Daniel T. Gryko et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Oxidative Cross-Coupling of Unfunctionalized Aromatic Compounds

(2009) Yasuyuki Kita et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cp2Ni-KOt-Bu-BEt3(or PPh3) Catalyst System for Direct C−H Arylation of Benzene, Naphthalene, and Pyridine

(2009) Osamu Kobayashi et al.   ORGANIC LETTERS

Copper-Mediated Direct Arylation of 1,3,4-Oxadiazoles and 1,2,4-Triazoles with Aryl Iodides

(2009) Tsuyoshi Kawano et al.   ORGANIC LETTERS

Nickel-Catalyzed Direct Arylation of Azoles with Aryl Bromides

(2009) Hitoshi Hachiya et al.   ORGANIC LETTERS

Practical Aspects of Carbon−Carbon Cross-Coupling Reactions Using Heteroarenes

(2009) Vincent F. Slagt et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed C−H Bond Activation

(2008) Jared C. Lewis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of 2-Arylbenzoxazoles by Copper-Catalyzed Intramolecular Oxidative CO Coupling of Benzanilides

(2008) Satoshi Ueda et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

CH Functionalization/CN Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

(2008) Gordon Brasche et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Coupling of Nitrogen Heteroaromatics and Alkanes without Transition Metals: A New Oxidative Cross-Coupling at CH/CH Bonds

(2008) Guojun Deng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Iron(III) Chloride Catalyzed Oxidative Coupling of Aromatic Nuclei

(2008) Kailiang Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Arylation and Alkenylation of Polyfluoroarene C−H Bonds

(2008) Hien-Quang Do et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Aerobic Oxidative Amidation of Terminal Alkynes:  Efficient Synthesis of Ynamides

(2008) Tetsuya Hamada et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rh(I)-Catalyzed Arylation of Heterocycles via C−H Bond Activation:  Expanded Scope through Mechanistic Insight

(2008) Jared C. Lewis et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(II)-Catalyzed Direct and Site-Selective Arylation of Indoles Under Mild Conditions

(2008) Robert J. Phipps et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Potassiumt-Butoxide Alone Can Promote the Biaryl Coupling of Electron-Deficient Nitrogen Heterocycles and Haloarenes

(2008) Shuichi Yanagisawa et al.   ORGANIC LETTERS

Oxidant-controlled regioselectivity in the oxidative arylation of N-acetylindoles

(2008) Shathaverdhan Potavathri et al.   TETRAHEDRON LETTERS

Copper-mediated direct arylation of benzoazoles with aryl iodides

(2008) Tomoki Yoshizumi et al.   TETRAHEDRON LETTERS

A general gold-catalyzed direct oxidative coupling of non-activated arenes

(2007) Anirban Kar et al.   CHEMICAL COMMUNICATIONS