An intramolecular tryptophan-condensation approach for peptide stapling

Orthogonal ring-closing alkyne and olefin metathesis for the synthesis of small GTPase-targeting bicyclic peptides

(2016) Philipp M. Cromm et al.   Nature Communications

Clinical Overview of MDM2/X-Targeted Therapies

(2016) Andrew Burgess et al.   Frontiers in Oncology

Double Strain-Promoted Macrocyclization for the Rapid Selection of Cell-Active Stapled Peptides

(2015) Yu Heng Lau et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Macrocyclization Reactions: The Importance of Conformational, Configurational, and Template-Induced Preorganization

(2015) Vicente Martí-Centelles et al.   CHEMICAL REVIEWS

Sensing Protein Surfaces with Targeted Fluorescent Receptors

(2015) Yael Nissinkorn et al.   CHEMISTRY-A EUROPEAN JOURNAL

Trp-Trp Cross-Linking: A Structure–Reactivity Relationship in the Formation and Design of Hyperstable Peptide β-Hairpin and α-Helix Scaffolds

(2015) Kamlesh M. Makwana et al.   ORGANIC LETTERS

Protein recognition by bivalent, ‘turn-on’ fluorescent molecular probes

(2015) Linor Unger-Angel et al.   Chemical Science

New peptide architectures through C–H activation stapling between tryptophan–phenylalanine/tyrosine residues

(2015) Lorena Mendive-Tapia et al.   Nature Communications

Diaminodiacid-Based Solid-Phase Synthesis of Peptide Disulfide Bond Mimics

(2013) Hong-Kui Cui et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Authorizing Multiple Chemical Passwords by a Combinatorial Molecular Keypad Lock

(2013) Bhimsen Rout et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Template-constrained macrocyclic peptides prepared from native, unprotected precursors

(2013) K. V. Lawson et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Stapled Peptides with Improved Potency and Specificity That Activate p53

(2012) Christopher J. Brown et al.   ACS Chemical Biology

Medication Detection by a Combinatorial Fluorescent Molecular Sensor

(2012) Bhimsen Rout et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

7,7′-Diamino-2,2′-diindolylmethane: A Building Block for Highly Efficient and Selective Anion Receptors-Studies in Solution and in the Solid State

(2012) Paweł Dydio et al.   CHEMISTRY-A EUROPEAN JOURNAL

Structure of the Stapled p53 Peptide Bound to Mdm2

(2011) Sohee Baek et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Selective fluorescent probes for live-cell monitoring of sulphide

(2011) Yong Qian et al.   Nature Communications

Hydrocarbon double-stapling remedies the proteolytic instability of a lengthy peptide therapeutic

(2010) G. H. Bird et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA