Temperature-modulated diastereoselective transformations of 2-vinylindoles to tetrahydrocarbazoles and tetrahydrocycloheptadiindoles

2- and 3-Vinylindoles as 4π Components in Cycloaddition Reactions

(2017) Elisabetta Rossi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Synthetic Route to Chiral 1,4-Disubstituted Tetrahydro-β-Carbolines via Domino Ring-Opening Cyclization of Activated Aziridines with 2-Vinylindoles

(2017) Masthanvali Sayyad et al.   JOURNAL OF ORGANIC CHEMISTRY

Construction of Chiral Tricyclic Indoles through a Rhodium-Catalyzed Asymmetric Arylation Protocol

(2017) Chun-Yan Wu et al.   ORGANIC LETTERS

[3 + 3] Cycloaddition of in Situ Formed Azaoxyallyl Cations with 2-Alkenylindoles: An Approach to Tetrahydro-β-carbolinones

(2017) Kaifan Zhang et al.   ORGANIC LETTERS

Syntheses of Tetrahydrobenzoazepinoindoles and Dihydrobenzodiazepinoindoles via Ring-Opening Cyclization of Activated Aziridines with 2-(2-Bromophenyl)-1H-indoles

(2017) Sajan Pradhan et al.   ORGANIC LETTERS

Diastereo- and enantioselective construction of biologically important pyrrolo[1,2-a]indole scaffolds via catalytic asymmetric [3 + 2] cyclodimerizations of 3-alkyl-2-vinylindoles

(2017) Zi-Qi Zhu et al.   Organic Chemistry Frontiers

Brønsted Acid-Catalyzed [3+2] Cyclodimerization of 3-Alkyl- 2-vinylindoles Leading to the Diastereoselective Construction of a Pyrroloindole Framework

(2016) Lei Yin et al.   ADVANCED SYNTHESIS & CATALYSIS

Gold(I)-Catalyzed Synthesis of Tetrahydrocarbazoles via Cascade [3,3]-Propargylic Rearrangement/[4+2] Cycloaddition of Vinylindoles and Propargylic Esters

(2016) Valentina Pirovano et al.   ADVANCED SYNTHESIS & CATALYSIS

Silver catalyzed domino aza-annulation/Diels–Alder cyclization of 2-ene-yne anilines: a facile one-pot access to carbazole, dihydrocarbazole and tetrahydrocarbazole frameworks

(2016) Namballa Hari Krishna et al.   CHEMICAL COMMUNICATIONS

Acid-Relayed Organocatalyticexo-Diels-Alder Cycloaddition of Cyclic Enones with 2-Vinyl-1H-indoles

(2016) Ji-Wei Ren et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Development and Scope of the Arene-Fused Domino Michael/Mannich Reaction: Application to the Total Syntheses of Aspidosperma Alkaloids (−)-Aspidospermidine, (−)-Tabersonine, and (−)-Vincadifformine

(2016) Senzhi Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

A Synthetic Route to Chiral Tetrahydropyrroloindoles via Ring Opening of Activated Aziridines with 2-Bromoindoles Followed by Copper-Catalyzed C–N Cyclization

(2016) Masthanvali Sayyad et al.   JOURNAL OF ORGANIC CHEMISTRY

Domino Ring-Opening Cyclization of Activated Aziridines with Indoles: Synthesis of Chiral Hexahydropyrroloindoles

(2016) Abhijit Mal et al.   JOURNAL OF ORGANIC CHEMISTRY

A Raney Cobalt Mediated Reductive Cyclization Route to the Uleine Alkaloid Gilbertine

(2016) Fei Tang et al.   JOURNAL OF ORGANIC CHEMISTRY

Exploiting the σ-phylic properties of cationic gold(i) catalysts in the ring opening reactions of aziridines with indoles

(2016) Elisabetta Rossi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective Construction of Functionalized Tetrahydrocarbazoles Enabled by Asymmetric Relay Catalysis of Gold Complex and Chiral Brønsted Acid

(2016) Feng Zhao et al.   ORGANIC LETTERS

Catalytic Enantioselective Synthesis of Tetrahydocarbazoles and Exocyclic Pictet–Spengler-Type Reactions

(2016) Casper L. Hansen et al.   ORGANIC LETTERS

Synthesis of constrained analogues of tryptophan

(2015) Elisabetta Rossi et al.   Beilstein Journal of Organic Chemistry

Catalytic Asymmetric Reactions of 4-Substituted Indoles with Nitroethene: A Direct Entry to Ergot Alkaloid Structures

(2015) Simone Romanini et al.   CHEMISTRY-A EUROPEAN JOURNAL

Brønsted Acid Catalyzed Asymmetric Diels–Alder Reactions: Stereoselective Construction of Spiro[tetrahydrocarbazole-3,3′-oxindole] Framework

(2015) Yang Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Construction of Benzo[c]carbazoles and Their Antitumor Derivatives through the Diels–Alder Reaction of 2-Alkenylindoles and Arynes

(2015) Feng Sha et al.   JOURNAL OF ORGANIC CHEMISTRY

One-Pot Catalytic Asymmetric Synthesis of Tetrahydrocarbazoles

(2015) Qiong-Jie Liu et al.   ORGANIC LETTERS

The asymmetric Cu(ii)–indolinylmethanol complex catalyzed Diels–Alder reaction of 2-vinylindoles with β,γ-unsaturated α-ketoesters: an efficient route to functionalized tetrahydrocarbazoles

(2014) Banlai Ouyang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Diastereoselective Synthesis of Functionalized Tetrahydrocarbazoles via a Domino-Ring Opening–Cyclization of Donor–Acceptor Cyclopropanes with Substituted 2-Vinylindoles

(2014) Ranadeep Talukdar et al.   ORGANIC LETTERS

Gold-catalyzed synthesis of tetrahydrocarbazole derivatives through an intermolecular cycloaddition of vinyl indoles and N-allenamides

(2013) Valentina Pirovano et al.   CHEMICAL COMMUNICATIONS

Intramolecular donor–acceptor cyclopropane ring-opening cyclizations

(2013) Marchello A. Cavitt et al.   CHEMICAL SOCIETY REVIEWS

Total Syntheses of the Monoterpene Indole Alkaloids (±)-Alstilobanine A and E and (±)-Angustilodine

(2013) Yiqing Feng et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Indole Substituted Twistenediones from a 2-Quinonyl Boronic Acid

(2013) Jaime Rojas-Martín et al.   ORGANIC LETTERS

Formal and total synthesis of (±)-cycloclavine

(2013) Nitinkumar D. Jabre et al.   TETRAHEDRON LETTERS

Total Synthesis of the Unusual Monoterpenoid Indole Alkaloid (±)-Alstilobanine A

(2012) Yiqing Feng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Occurrence, Biogenesis, and Synthesis of Biologically Active Carbazole Alkaloids

(2012) Arndt W. Schmidt et al.   CHEMICAL REVIEWS

Protecting-Group-Free Total Synthesis of (E)- and (Z)-Alstoscholarine

(2011) Thibaud Gerfaud et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of (±)-Cycloclavine and (±)-5-epi-Cycloclavine

(2011) Filip R. Petronijevic et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Biomimetic Total Syntheses of Flinderoles B and C

(2011) Dattatraya H. Dethe et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A new procedure for the preparation of 2-vinylindoles and their [4+2] cycloaddition reaction

(2011) Yaseen Ali Mosa Mohamed et al.   TETRAHEDRON

An Enantioselective Approach to Highly Substituted Tetrahydrocarbazoles through Hydrogen Bonding-Catalyzed Cascade Reactions

(2010) Xu-Fan Wang et al.   ORGANIC LETTERS

Brønsted acid catalyzed Diels–Alder reactions of 2-vinylindoles and 3-nitrocoumarins: an expedient synthesis of coumarin-fused tetrahydrocarbazoles

(2010) Fen Tan et al.   TETRAHEDRON

Structure−Activity Relationship Studies Leading to the Identification of (2E)-3-[l-[(2,4-Dichlorophenyl)methyl]-5-fluoro-3-methyl-lH-indol-7-yl]-N-[(4,5-dichloro-2-thienyl)sulfonyl]-2-propenamide (DG-041), a Potent and Selective Prostanoid EP3 Receptor Antagonist, as a Novel Antiplatelet Agent That Does Not Prolong Bleeding

(2009) Jasbir Singh et al.   JOURNAL OF MEDICINAL CHEMISTRY

Brønsted Acid Mediated Tandem Diels−Alder/Aromatization Reactions of Vinylindoles

(2009) Cai-Bao Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Protecting-group-free synthesis as an opportunity for invention

(2009) Ian S. Young et al.   Nature Chemistry

New routes to clavine-type ergot alkaloids. Part 2: Synthesis of the last, so far not yet synthesized member of the clavine alkaloid family, (±)-cycloclavine

(2008) Mária Incze et al.   TETRAHEDRON