Journal
JOURNAL OF ORGANIC CHEMISTRY
Volume 83, Issue 8, Pages 4641-4649Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.8b00388
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Funding
- National Research Foundation of Korea (NRF) - Korea government (MSIP) [2016R1A4A1011189, 2017R1D1A1A09000574, 2017R1A2B2004786]
- National Research Foundation of Korea [2017R1A2B2004786, 2017R1D1A1A09000574] Funding Source: Korea Institute of Science & Technology Information (KISTI), National Science & Technology Information Service (NTIS)
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The ruthenium(II)-catalyzed C-H aminocarbonylation of N-(hetero)aryl-7-azaindoles with isocyanates is described. The excellent site selectivity at the ortho-position within the N-(hetero)aryl ring was observed to provide ortho-amidated N-(hetero)aryl-7-azaindoles under the mild reaction conditions. The resulting 7-azaindole derivatives can be readily transformed into 7-azaindoles containing carboxylic acid and alkyl amine functional groups.
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