Anti-inflammatory Exploration of Sulfonamide Containing Diaryl Pyrazoles with Promising COX-2 Selectivity and Enhanced Gastric Safety Profile

Design, synthesis and biological screening of new 4-thiazolidinone derivatives with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile

(2016) Khaled R.A. Abdellatif et al.   BIOORGANIC CHEMISTRY

The therapeutic voyage of pyrazole and its analogs: A review

(2016) Mohemmed Faraz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and anticancer activities of novel (tetrahydrobenzo [4,5] thieno [2,3-d] pyrimidine-4-yl)-pyrolidine-2-carboxylic acid derivatives

(2016) Laxmikant S. Pavase et al.   MEDICINAL CHEMISTRY RESEARCH

Design, synthesis, and biological evaluation of novel fluorinated pyrazole encompassing pyridyl 1,3,4-oxadiazole motifs

(2016) Nisheeth C. Desai et al.   MEDICINAL CHEMISTRY RESEARCH

Evaluation of anti-inflammatory, analgesic activities, and side effects of some pyrazole derivatives

(2016) Souraya Domiati et al.   INFLAMMOPHARMACOLOGY

Celecoxib analogs bearing benzofuran moiety as cyclooxygenase-2 inhibitors: Design, synthesis and evaluation as potential anti-inflammatory agents

(2014) Ghaneya Sayed Hassan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Novel 3-substituted-1-aryl-5-phenyl-6-anilinopyrazolo[3,4-d]pyrimidin-4-ones: Docking, synthesis and pharmacological evaluation as a potential anti-inflammatory agents

(2012) Sandeep B. Yewale et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors

(2011) Baker Jawabrah Al-Hourani et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of pyrazole derivatives containing thiourea skeleton as anticancer agents

(2010) Peng-Cheng Lv et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The novel benzopyran class of selective cyclooxygenase-2 inhibitors. Part 2: The second clinical candidate having a shorter and favorable human half-life

(2010) Jane L. Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and antimicrobial activity of some new thiazole, thiophene and pyrazole derivatives containing benzothiazole moiety

(2010) Samir Bondock et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design and synthesis of new 1,3-benzthiazinan-4-one derivatives as selective cyclooxygenase (COX-2) inhibitors

(2009) Afshin Zarghi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of 3-alkyl-2-aryl-1,3-thiazinan-4-one derivatives as selective cyclooxygenase (COX-2) inhibitors

(2009) Tannaz Zebardast et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of novel pyrazole derivatives and evaluation of their antidepressant and anticonvulsant activities

(2009) Mohamed Abdel-Aziz et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide

(2008) I.G. Rathish et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS