Synthesis of triazolylmethyl-linked nucleoside analogs via combination of azidofuranoses with propargylated nucleobases and study on their cytotoxicity

Synthesis and antimicrobial evaluation of sulfanilamide- and carbohydrate-derived 1,4-disubstitued-1,2,3-triazoles via click chemistry

(2017) Kadir Ay et al.   MEDICINAL CHEMISTRY RESEARCH

Synthesis of Rapamycin Derivatives Containing the Triazole Moiety Used as Potential mTOR-Targeted Anticancer Agents

(2016) Lijun Xie et al.   ARCHIV DER PHARMAZIE

Click-based synthesis and antitubercular evaluation of novel dibenzo[ b , d ]thiophene-1,2,3-triazoles with piperidine, piperazine, morpholine and thiomorpholine appendages

(2016) Lokesh Pulipati et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Application of the Huisgen cycloaddition and ‘click’ reaction toward various 1,2,3-triazoles as HIV non-nucleoside reverse transcriptase inhibitors

(2016) Nicole Pribut et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Seeking potent anti-tubercular agents: Design, synthesis, anti-tubercular activity and docking study of various ((triazoles/indole)-piperazin-1-yl/1,4-diazepan-1-yl)benzo[d]isoxazole derivatives

(2016) Kalaga Mahalakshmi Naidu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and cytotoxic evaluation of novel indenoisoquinoline-substituted triazole hybrids

(2016) Tham Pham Thi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery of novel pyrrolo[2,3-b]pyridine derivatives bearing 1,2,3-triazole moiety as c-Met kinase inhibitors

(2016) Qidong Tang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cu-Catalyzed Click Reaction in Carbohydrate Chemistry

(2016) Vinod K. Tiwari et al.   CHEMICAL REVIEWS

Synthesis of newer 1,2,3-triazole linked chalcone and flavone hybrid compounds and evaluation of their antimicrobial and cytotoxic activities

(2016) Rama Kant et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of Novel Triazole-incorporated Isatin Derivatives as Antifungal, Antitubercular, and Antioxidant Agents and Molecular Docking Study

(2016) Mubarak H. Shaikh et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

9H-Carbazole Derivatives Containing theN-Benzyl-1,2,3-triazole Moiety as New Acetylcholinesterase Inhibitors

(2015) Hamidreza Akrami et al.   ARCHIV DER PHARMAZIE

New carbocyclic N6-substituted adenine and pyrimidine nucleoside analogues with a bicyclo[2.2.1]heptane fragment as sugar moiety; synthesis, antiviral, anticancer activity and X-ray crystallography

(2015) Constantin I. Tănase et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of 1,2-benzisoxazole tethered 1,2,3-triazoles that exhibit anticancer activity in acute myeloid leukemia cell lines by inhibiting histone deacetylases, and inducing p21 and tubulin acetylation

(2015) Nanjundaswamy Ashwini et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Deprotometalation–iodolysis and computed CH acidity of 1,2,3- and 1,2,4-triazoles. Application to the synthesis of resveratrol analogues

(2015) Elisabeth Nagaradja et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Click reaction based synthesis, antimicrobial, and cytotoxic activities of new 1,2,3-triazoles

(2015) Mohamed Ramadan El Sayed Aly et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design and synthesis of novel 1,2,3-triazole–pyrimidine–urea hybrids as potential anticancer agents

(2015) Li-Ying Ma et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Mechanochemical click reaction as a tool for making carbohydrate-based triazole-linked self-assembling materials (CTSAMs)

(2015) Mohit Tyagi et al.   CARBOHYDRATE RESEARCH

Synthesis of 1,2,3-triazole-linked glycohybrids in the gluco-, gulo-, and allopyranose series

(2015) Jevgeņija Uzuleņa et al.   Chemistry of Heterocyclic Compounds

Synthesis of purine and 2-aminopurine conjugates bearing the fragments of heterocyclic amines at position 6

(2015) Dmitry A. Gruzdev et al.   Chemistry of Heterocyclic Compounds

Synthesis of monomeric methylene-linked 1,2,3-triazole glycoconjugates from allo- and glucofuranoses

(2015) Jeļena Grigorjeva et al.   Chemistry of Heterocyclic Compounds

Semi-Synthesis of new glycosidic triazole derivatives of dihydrocucurbitacin B

(2015) Ana L.M. Morotti et al.   TETRAHEDRON LETTERS

Novel Acyclic Phosphonylated 1,2,3-Triazolonucleosides with an Acetamidomethyl Linker: Synthesis and Biological Activity

(2014) Iwona E. Głowacka et al.   ARCHIV DER PHARMAZIE

Synthesis of novel pyrimidine nucleoside analogues owning multiple bases/sugars and their glycosidase inhibitory activity

(2014) Ravi Kumar Thakur et al.   TETRAHEDRON

Design, synthesis, and biological evaluation of new 2′-deoxy-2′-fluoro-4′-triazole cytidine nucleosides as potent antiviral agents

(2013) Jie Wu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Advances in the development of nucleoside and nucleotide analogues for cancer and viral diseases

(2013) Lars Petter Jordheim et al.   NATURE REVIEWS DRUG DISCOVERY

The Newest Member of the Family of Chloralose: Synthesis ofβ-Ribochloralose and Some Derivatives

(2013) Kadir Ay et al.   Journal of Chemistry

Semi-Synthesis and Biological Evaluation of 1,2,3-Triazole-Based Podophyllotoxin Congeners as Potent Antitumor Agents Inducing Apoptosis in HepG2 Cells

(2012) Jinying Chen et al.   ARCHIV DER PHARMAZIE

Triazole pyrimidine nucleosides as inhibitors of Ribonuclease A. Synthesis, biochemical, and structural evaluation

(2012) Vanessa Parmenopoulou et al.   BIOORGANIC & MEDICINAL CHEMISTRY

New triazole derivatives as antifungal agents: Synthesis via click reaction, in vitro evaluation and molecular docking studies

(2012) Yan Zou et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of 1,2,3-triazole glycoconjugates as inhibitors of α-glucosidases

(2012) David R. da Rocha et al.   CARBOHYDRATE RESEARCH

Catalytic Stereoselective Synthesis of Diverse Oxindoles and Spirooxindoles from Isatins

(2012) Jacob P. MacDonald et al.   ACS Combinatorial Science

In vitro and QSAR studies of cucurbitacins on HepG2 and HSC-T6 liver cell lines

(2011) Judit Bartalis et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design, synthesis and the effect of 1,2,3-triazole sialylmimetic neoglycoconjugates on Trypanosoma cruzi and its cell surface trans-sialidase

(2011) Vanessa L. Campo et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Click Chemistry: 1,2,3-Triazoles as Pharmacophores

(2011) Sandip G. Agalave et al.   Chemistry-An Asian Journal

Synthesis and antiviral evaluation of 1,3-dimethyl-6-(1H-1,2,3-triazol-1-YL)pyrimidine-2,4(1H,3H)-dione derivatives

(2010) A. Sh. El-Etrawy et al.   Chemistry of Heterocyclic Compounds

Synthesis, Biological Activity, and Molecular Modeling Studies of 1H-1,2,3-Triazole Derivatives of Carbohydrates as α-Glucosidases Inhibitors

(2010) Sabrina B. Ferreira et al.   JOURNAL OF MEDICINAL CHEMISTRY

2-Aryl-3-(1H-Azol-1-yl)-1H-Indole Derivatives: A New Class of Antimycobacterial Compounds – Conventional Heating in Comparison with MW-Assisted Synthesis

(2009) Daniele Zampieri et al.   ARCHIV DER PHARMAZIE

Nucleosides and oligonucleotides containing 1,2,3-triazole residues with nucleobase tethers: Synthesis via the azide-alkyne ‘click’ reaction

(2008) Padmaja Chittepu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, HIV-RT inhibitory activity and SAR of 1-benzyl-1H-1,2,3-triazole derivatives of carbohydrates

(2008) Fernando de C. da Silva et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY