Identification of inhibitors of Tartrate-resistant acid phosphatase (TRAP/ACP5 ) activity by small-molecule screening

A Potent Tartrate Resistant Acid Phosphatase Inhibitor to Study the Function of TRAP in Alveolar Macrophages

(2017) Carian E. Boorsma et al.   Scientific Reports

Identification of Drug-Like Inhibitors of Insulin-Regulated Aminopeptidase Through Small-Molecule Screening

(2016) Karin Engen et al.   ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES

Tartrate-Resistant Acid Phosphatase Deficiency in the Predisposition to Systemic Lupus Erythematosus

(2016) Jie An et al.   Arthritis & Rheumatology

The small chemical enzyme inhibitor 5-phenylnicotinic acid/CD13 inhibits cell migration and invasion of tartrate-resistant acid phosphatase/ACP5-overexpressing MDA-MB-231 breast cancer cells

(2015) Michael Krumpel et al.   EXPERIMENTAL CELL RESEARCH

An Aggregation Advisor for Ligand Discovery

(2015) John J. Irwin et al.   JOURNAL OF MEDICINAL CHEMISTRY

Terpenes and sterols from the fruits of Prunus mume and their inhibitory effects on osteoclast differentiation by suppressing tartrate-resistant acid phosphatase activity

(2014) Xi-Tao Yan et al.   ARCHIVES OF PHARMACAL RESEARCH

Increased Tartrate-Resistant Acid Phosphatase Expression in Osteoblasts and Osteocytes in Experimental Osteoporosis in Rats

(2014) Lene B. Solberg et al.   CALCIFIED TISSUE INTERNATIONAL

ACP5, a direct transcriptional target of FoxM1, promotes tumor metastasis and indicates poor prognosis in hepatocellular carcinoma

(2013) L Xia et al.   ONCOGENE

Polyphosphate-Mediated Inhibition of Tartrate-Resistant Acid Phosphatase and Suppression of Bone Resorption of Osteoclasts

(2013) Kana Harada et al.   PLoS One

Identification of Purple Acid Phosphatase Inhibitors by Fragment-Based Screening: Promising New Leads for Osteoporosis Therapeutics

(2012) Daniel Feder et al.   Chemical Biology & Drug Design

A consistent description of HYdrogen bond and DEhydration energies in protein–ligand complexes: methods behind the HYDE scoring function

(2012) Nadine Schneider et al.   JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN

Synthesis, modelling and kinetic assays of potent inhibitors of purple acid phosphatase

(2011) Siti Hajar Mohd-Pahmi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Proinvasion Metastasis Drivers in Early-Stage Melanoma Are Oncogenes

(2011) Kenneth L. Scott et al.   CANCER CELL

Expression and secretion of the novel adipokine tartrate-resistant acid phosphatase from adipose tissues of obese and lean women

(2011) P Lång et al.   INTERNATIONAL JOURNAL OF OBESITY

Biogenesis of tartrate-resistant acid phosphatase isoforms 5a and 5b in stably transfected MDA-MB-231 breast cancer epithelial cells

(2010) Serhan Zenger et al.   BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH

Tartrate-resistant acid phosphatase isoform 5b (TRACP 5b) as a serum maker for cancer with bone metastasis

(2010) Tsu-Yi Chao et al.   CLINICA CHIMICA ACTA

Serum tartrate-resistant acid phosphatase 5b (TRACP5b) activity as a biomarker for bone metastasis in non-small cell lung cancer patients

(2010) Nai-Shun Yao et al.   CLINICA CHIMICA ACTA

Differential expression of tartrate-resistant acid phosphatase isoforms 5a and 5b by tumor and stromal cells in human metastatic bone disease

(2010) Serhan Zenger et al.   CLINICAL & EXPERIMENTAL METASTASIS

Apparent activity in high-throughput screening: origins of compound-dependent assay interference

(2010) Natasha Thorne et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Tartrate-resistant acid phosphatase from human bone: Purification and development of an immunoassay

(2010) Jussi Halleen et al.   JOURNAL OF BONE AND MINERAL RESEARCH

Inhibition of purple acid phosphatase with α-alkoxynaphthylmethylphosphonic acids

(2008) Ross P. McGeary et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Gold(III) compounds as anticancer agents: Relevance of gold–protein interactions for their mechanism of action

(2007) Angela Casini et al.   JOURNAL OF INORGANIC BIOCHEMISTRY