Synthesis and biological evaluation of novel N -aryl-ω -(benzoazol-2-yl)-sulfanylalkanamides as dual inhibitors of α-glucosidase and protein tyrosine phosphatase 1B

Inhibitory mechanism of two allosteric inhibitors, oleanolic acid and ursolic acid on α-glucosidase

(2018) Huafang Ding et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Inhibitory activity evaluation and mechanistic studies of tetracyclic oxindole derivatives as α-glucosidase inhibitors

(2016) Hua Sun et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Protein tyrosine phosphatase 1B and α-glucosidase inhibitory activities of Pueraria lobata root and its constituents

(2016) Su Hui Seong et al.   JOURNAL OF ETHNOPHARMACOLOGY

Design, synthesis and docking study of novel tetracyclic oxindole derivatives as α-glucosidase inhibitors

(2015) Kailin Han et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, biological evaluation and 3D-QSAR studies of imidazolidine-2,4-dione derivatives as novel protein tyrosine phosphatase 1B inhibitors

(2015) Mei-Yan Wang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of novel flavone hydrazones: In-vitro evaluation of α-glucosidase inhibition, QSAR analysis and docking studies

(2015) Syahrul Imran et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Chemical Constituents ofEuonymus alatus(Thunb.) Sieb. and Their PTP1B and α-Glucosidase Inhibitory Activities

(2015) Su-Yang Jeong et al.   PHYTOTHERAPY RESEARCH

Sulfur rich 2-mercaptobenzothiazole and 1,2,3-triazole conjugates as novel antitubercular agents

(2014) Fauzia Mir et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Xanthohumol, a Prenylated Chalcone from Beer Hops, Acts as an α-Glucosidase Inhibitor in Vitro

(2014) Ming Liu et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

2-(2-Arylphenyl)benzoxazole As a Novel Anti-Inflammatory Scaffold: Synthesis and Biological Evaluation

(2014) Kapileswar Seth et al.   ACS Medicinal Chemistry Letters

Design, synthesis and molecular modelling studies of novel 3-acetamido-4-methyl benzoic acid derivatives as inhibitors of protein tyrosine phosphatase 1B

(2013) Monika Rakse et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Development of a Chimeric c-Src Kinase and HDAC Inhibitor

(2013) Kristin S. Ko et al.   ACS Medicinal Chemistry Letters

Molecular modeling and synthesis of ZINC02765569 derivatives as protein tyrosine phosphatase 1B inhibitors: lead optimization study

(2012) Prashant Joshi et al.   MEDICINAL CHEMISTRY RESEARCH

Automated design of ligands to polypharmacological profiles

(2012) Jérémy Besnard et al.   NATURE

SYNTHESIS AND EVALUATION OF 5-(6-METHOXYNAPHTHALEN-2-YL)-1-ARYL-1-(4-(TRIFLUOROMETHYL)PHENYLAMINO)PENTAN-3-ONE AS POTENTIAL ANTIDIABETIC AGENTS

(2012) HAN HAI YAN et al.   JOURNAL OF THE CHILEAN CHEMICAL SOCIETY

Synthesis, DNA-binding ability and anticancer activity of benzothiazole/benzoxazole–pyrrolo[2,1-c][1,4]benzodiazepine conjugates

(2010) Ahmed Kamal et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity

(2010) Deju Ye et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Efficacy and safety of a selective estrogen receptor β agonist, ERB-041, in patients with rheumatoid arthritis: A 12-week, randomized, placebo-controlled, phase II study

(2010) Jorge A. Roman-Blas et al.   ARTHRITIS CARE & RESEARCH

Discovery of a novel competitive inhibitor of PTP1B by high-throughput screening

(2008) Lei SHI et al.   ACTA PHARMACOLOGICA SINICA

Oleanolic acid and its derivatives: New inhibitor of protein tyrosine phosphatase 1B with cellular activities

(2008) Yi-Nan Zhang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Preparation and in vitro evaluation of benzylsulfanyl benzoxazole derivatives as potential antituberculosis agents

(2008) Věra Klimešová et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Antioxidant constituents in the dayflower (Commelina communis L.) and their α-glucosidase-inhibitory activity

(2008) Makio Shibano et al.   Journal of Natural Medicines