Synthesis and pharmacological evaluation of 2,3-diphenyl acrylonitriles-bearing halogen as selective anticancer agents

Synthesis and evaluation of a radioiodinated 4,6-diaryl-3-cyano-2-pyridinone derivative as a survivin targeting SPECT probe for tumor imaging

(2016) Takeshi Fuchigami et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Syntheses and biological evaluation of 1,2,3-triazole and 1,3,4-oxadiazole derivatives of imatinib

(2016) Yong-Tao Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

New small molecule inhibitors of histone methyl transferase DOT1L with a nitrile as a non-traditional replacement for heavy halogen atoms

(2016) Sophie S. Spurr et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological activity of pyrrole analogues of combretastatin A-4

(2016) Eun-Kyung Jung et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

New ( E )-1-alkyl-1 H -benzo[ d ]imidazol-2-yl)methylene)indolin-2-ones: Synthesis, in vitro cytotoxicity evaluation and apoptosis inducing studies

(2016) Pankaj Sharma et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Combretastatins: In vitro structure-activity relationship, mode of action and current clinical status

(2016) Karol Jaroch et al.   Pharmacological Reports

Synthesis andIn VitroActivity of Polyhalogenated 2-phenylbenzimidazoles as a New Class of anti-MRSA and Anti-VRE Agents

(2015) Hakan Göker et al.   Chemical Biology & Drug Design

Synthesis and biological evaluation of novel 4,5-disubstituted 2H-1,2,3-triazoles as cis-constrained analogues of combretastatin A-4

(2015) Nikhil R. Madadi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Partial Convergence in Action of Methylene Blue and Artemisinins: Antagonism with Chloroquine, a Reversal with Verapamil, and an Insight into the Antimalarial Activity of Chloroquine

(2011) Richard K. Haynes et al.   ChemMedChem

Rho-associated kinase (ROCK) inhibition reverses low cell activity on hydrophobic surfaces

(2009) Yu Shun Tian et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS