Journal
JOURNAL OF ORGANIC CHEMISTRY
Volume 82, Issue 5, Pages 2764-2771Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.7b00002
Keywords
-
Categories
Funding
- CSIR New Delhi [02(0212)/14/EMR.-II]
- UGC New Delhi
Ask authors/readers for more resources
A copper-catalyzed selective C-N cross-coupling has been developed based on chelation-assisted amidation of readily available aryl boronic acids at room-temperature under open-flask conditions. The reaction is scalable and tolerates a wide spectrum of functional groups delivering fully substituted unsymmetrical amides in high yields (up to 96%). The C-N cross coupling also established with aryl silanes, extending the palette of coupling partners of this strategy.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available