Journal
JOURNAL OF ORGANIC CHEMISTRY
Volume 82, Issue 4, Pages 2081-2088Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.6b02906
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Funding
- National Natural Science Foundation of China [21172001, 21372008]
- Natural Science Foundation of Education Administration of Anhui Province [KJ2016A267]
- Special and Excellent Research Fund of Anhui Normal University
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A mild and efficient Rh(III)-catalyzed C-H activation/esterification reaction for the synthesis of isocoumarins has been developed. This procedure uses readily available benzoic acids and cyclic diazo-1,3-diketones as starting materials and involves domino intermolecular C-H activation in combination with intramolecular esterification to give the corresponding isocoumarins in moderate to excellent yields. This process provides a facile approach for the construction of isocoumarins containing various functional groups that does not require any additives.
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