Fast, solvent-free and highly enantioselective fluorination of β-keto esters catalyzed by chiral copper complexes in a ball mill

Reagent-controlled enantioselectivity switch for the asymmetric fluorination of β-ketocarbonyls by chiral primary amine catalysis

(2017) Yang'en You et al.   Chemical Science

Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas

(2016) Yu Zhou et al.   CHEMICAL REVIEWS

Fast, solvent-free, highly enantioselective three-component coupling of aldehydes, alkynes, and amines catalysed by the copper(ii)pybox complex under high-vibration ball-milling

(2015) Zhenhua Li et al.   GREEN CHEMISTRY

Metal-catalyzed organic reactions using mechanochemistry

(2015) José G. Hernández et al.   TETRAHEDRON LETTERS

Iron(iii)–salan complexes catalysed highly enantioselective fluorination and hydroxylation of β-keto esters and N-Boc oxindoles

(2014) Xin Gu et al.   CHEMICAL COMMUNICATIONS

Advances in Catalytic Enantioselective Fluorination, Mono-, Di-, and Trifluoromethylation, and Trifluoromethylthiolation Reactions

(2014) Xiaoyu Yang et al.   CHEMICAL REVIEWS

Mechanochemistry: a web themed issue

(2013) Stuart L. James et al.   CHEMICAL COMMUNICATIONS

Mechanochemical organic synthesis

(2013) Guan-Wu Wang   CHEMICAL SOCIETY REVIEWS

Enantioselective Fluorination of β-Ketoesters Catalyzed by Chiral Sodium Phosphate: Remarkable Enhancement of Reactivity by Simultaneous Utilization of Metal Enolate and Metal Phosphate

(2013) Keiji Mori et al.   CHEMISTRY LETTERS

Organocatalytic solvent-free hydrogen bonding-mediated asymmetric Michael additions under ball milling conditions

(2013) Manuel Jörres et al.   GREEN CHEMISTRY

Fast, solvent-free asymmetric alkynylation of prochiral sp3 C–H bonds in a ball mill for the preparation of optically active tetrahydroisoquinoline derivatives

(2013) Jingbo Yu et al.   TETRAHEDRON LETTERS

Enantioselective direct fluorination and chlorination of cyclic β-ketoesters mediated by phase-transfer catalysts

(2013) Jie Luo et al.   TETRAHEDRON LETTERS

Efficient enantioselective fluorination of β-keto esters/amides catalysed by diphenylamine-linked bis(thiazoline)–Cu(OTf)2complexes

(2013) Jiahuan Peng et al.   RSC Advances

Thiourea-Catalyzed Enantioselective Fluorination of β-Keto Esters

(2012) Junxing Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Asymmetric Mono-Fluorination of α-Keto Esters: Synthesis of Optically Active β-Fluoro-α-Hydroxy and β-Fluoro-α-Amino Acid Derivatives

(2012) Shoko Suzuki et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Mechanochemistry assisted asymmetric organocatalysis: A sustainable approach

(2012) Pankaj Chauhan et al.   Beilstein Journal of Organic Chemistry

Preparation of Chiral Amino Esters by Asymmetric Phase-Transfer Catalyzed Alkylations of Schiff Bases in a Ball Mill

(2012) Pierrick Nun et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fast, solvent-free and hydrogen-bonding-mediated asymmetric Michael addition in a ball mill

(2012) Yi-Feng Wang et al.   GREEN CHEMISTRY

Substrate Range of the Titanium TADDOLate Catalyzed Asymmetric Fluorination of Activated Carbonyl Compounds

(2012) Andreas Bertogg et al.   HELVETICA CHIMICA ACTA

Ball milling in organic synthesis: solutions and challenges

(2011) Achim Stolle et al.   CHEMICAL SOCIETY REVIEWS

Mechanochemistry: opportunities for new and cleaner synthesis

(2011) Stuart L. James et al.   CHEMICAL SOCIETY REVIEWS

Transition Metal Catalyzed Enantioselective α-Heterofunctionalization of Carbonyl Compounds

(2010) Alexander M. R. Smith et al.   CHEMICAL REVIEWS

Chiral bifunctional phase transfer catalysts for asymmetric fluorination of β-keto esters

(2009) Xisheng Wang et al.   CHEMICAL COMMUNICATIONS

Recent advances in the synthesis of fluorinated nucleosides

(2009) Xiao-Long Qiu et al.   TETRAHEDRON

Fluorination in Medicinal Chemistry: Methods, Strategies, and Recent Developments

(2008) Kenneth L. Kirk   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Desymmetrization-like Catalytic Enantioselective Fluorination of Malonates and Its Application to Pharmaceutically Attractive Molecules

(2007) Dhande Sudhakar Reddy et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Understanding organofluorine chemistry. An introduction to the C–F bond

(2007) David O'Hagan   CHEMICAL SOCIETY REVIEWS

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS