The Baldwin Rearrangement: Synthesis of 2-Acylaziridines

Solid-phase synthesis, cyclization, and site-specific functionalization of aziridine-containing tetrapeptides

(2017) Benjamin K W Chung et al.   Nature Protocols

Zinc Iodide-Mediated Direct Synthesis of 2,3-Dihydroisoxazoles from Alkynes and Nitrones

(2016) Zu-Feng Xiao et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Hydrogenation of Isoxazolium Triflates with a Chiral Iridium Catalyst

(2016) Ryuhei Ikeda et al.   CHEMISTRY-A EUROPEAN JOURNAL

Unexpected synthesis of aziridines under Cu(I) catalyzed Kinugasa conditions assisted by microwave irradiation

(2016) Heithem Abda et al.   COMPTES RENDUS CHIMIE

Synthesis of Some Novel Class of Bis(isoxazoline) and Bis(aziridine) Derivatives

(2016) Bhaskar Chakraborty et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Synthesis of 4-Isoxazolines through Gold(I)-Catalyzed Cyclization of Propargylic N-Hydroxylamines

(2016) B. Chandrasekhar et al.   JOURNAL OF ORGANIC CHEMISTRY

The effect of backbone flexibility on site-selective modification of macrocycles

(2016) Conor C. G. Scully et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Asymmetric Construction of 2,3-Dihydroisoxazoles via an Organocatalytic Formal [3 + 2] Cycloaddition of Enynes with N-Hydroxylamines

(2016) Wenbo Li et al.   ORGANIC LETTERS

The reactivity and conformational control of cyclic tetrapeptides derived from aziridine-containing amino acids

(2016) Benjamin K. W. Chung et al.   Chemical Science

Solid-Phase Parallel Synthesis of Functionalised Medium-to-Large Cyclic Peptidomimetics through Three-Component Coupling Driven by Aziridine Aldehyde Dimers

(2015) Adam P. Treder et al.   CHEMISTRY-A EUROPEAN JOURNAL

Highly Stereoselective Synthesis of New Aziridines via Baldwin Rearrangement and Their Potential Biological Activities

(2015) Bhaskar Chakraborty et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Diversity in Synthesis of N-Heterocycles from Simple Propargylic Alcohols

(2015) Emmanuel Vrancken et al.   SYNLETT

Mechanistic investigation of aziridine aldehyde-driven peptide macrocyclization: the imidoanhydride pathway

(2015) Serge Zaretsky et al.   Chemical Science

Synthesis and Reactivity of 2-(Carboxymethyl)aziridine Derivatives

(2014) Gert Callebaut et al.   CHEMICAL REVIEWS

Ruthenium Porphyrin Catalyzed Three-Component Reaction of Diazo Compounds, Nitrosoarenes, and Alkynes: An Efficient Approach to Multifunctionalized Aziridines

(2014) Annapureddy Rajasekar Reddy et al.   ORGANIC LETTERS

A Lewis acid/metal amide hybrid as an efficient catalyst for carbon–carbon bond formation

(2014) Yasuhiro Yamashita et al.   Chemical Science

Application of Regio- and Stereoselective Functional Group Transformations of Chiral Aziridine-2-carboxylates

(2014) Hyun-Joon Ha et al.   Asian Journal of Organic Chemistry

Mitomycinoid Alkaloids: Mechanism of Action, Biosynthesis, Total Syntheses, and Synthetic Approaches

(2013) Phillip D. Bass et al.   CHEMICAL REVIEWS

One-Pot Stereoselective Synthesis of 2-Acylaziridines and 2-Acylpyrrolidines fromN-(Propargylic)hydroxylamines

(2013) Yoshiaki Miyamoto et al.   Chemistry-An Asian Journal

Kinugasa Reaction: A Direct One-Pot Route to Highly Functionalized β-Lactams

(2013) Rama K. Khangarot et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

N-Alkoxyheterocycles As Irreversible Photooxidants

(2013) Zofia M. Wosinska et al.   PHOTOCHEMISTRY AND PHOTOBIOLOGY

A simple, efficient, regioselective and one-pot preparation of N-hydroxy- and N–O-protected hydroxyindoles via cycloaddition of nitrosoarenes with alkynes. Synthetic scope, applications and novel by-products

(2013) Gabriella Ieronimo et al.   TETRAHEDRON

A new route to the synthesis of isoxazoline derivatives from dihydropyran via cycloaddition reaction in ionic liquid

(2013) Bhaskar Chakraborty et al.   TETRAHEDRON LETTERS

Bicycle synthesis through peptide macrocyclization using aziridine aldehydes followed by late stage disulfide bond installation

(2013) Benjamin K. W. Chung et al.   MedChemComm

Novel achievements with an old metal: copper-promoted synthesis of four-membered azacycles

(2013) Benito Alcaide et al.   RSC Advances

Organocatalytic Enantioselective Dipolar [3+2] Cycloadditions of Acetylenic Aldehydes with Nitrones for the Formation of Chiral 4-Isoxazolines

(2012) Xianrong Cai et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Synthesis of 4-Isoxazolines by 1,3-Dipolar Cycloadditions of Nitrones to Alkynals Catalyzed by Fluorodiphenylmethylpyrrolidines

(2012) José Alemán et al.   ADVANCED SYNTHESIS & CATALYSIS

Conformational Modulation of in Vitro Activity of Cyclic RGD Peptides via Aziridine Aldehyde-Driven Macrocyclization Chemistry

(2012) Áron Roxin et al.   BIOCONJUGATE CHEMISTRY

Bending Rigid Molecular Rods: Formation of Oligoproline Macrocycles

(2012) Conor C. G. Scully et al.   CHEMISTRY-A EUROPEAN JOURNAL

DNA Interstrand Cross-Linking Agents and their Chemotherapeutic Potential

(2012) L. Brulikova et al.   CURRENT MEDICINAL CHEMISTRY

Aziridine-2-carboxylates: Preparation, Nucleophilic Ring Opening, and Ring Expansion

(2012) Tsutomu Ishikawa   HETEROCYCLES

Stereoselective Synthesis of 1-Nitrobicyclo[3.1.0]hexanes and Fused Isoxazoline-N-oxides from Primary Nitro Compounds

(2012) Akio Kamimura et al.   JOURNAL OF ORGANIC CHEMISTRY

A Versatile Scaffold for Site-Specific Modification of Cyclic Tetrapeptides

(2012) Christopher J. White et al.   ORGANIC LETTERS

Aziridine-2-carboxaldehyde Dimers Undergo Homo-Ugi 4-Component-5-center Reactions

(2012) Andrei Yudin et al.   SYNTHESIS-STUTTGART

Synthetic studies on pactamycin, a potent antitumor antibiotic

(2012) Nobuyuki Matsumoto et al.   RSC Advances

Regioselectivity in the ring opening of non-activated aziridines

(2011) Sonja Stanković et al.   CHEMICAL SOCIETY REVIEWS

Selective Transformation ofN-(Propargylic)hydroxylamines into 4-Isoxazolines and Acylaziridines Promoted by Metal Salts

(2011) Norihiro Wada et al.   CHEMISTRY LETTERS

Optically Active Bicyclic N-Heterocycles by Organocatalytic Asymmetric Michael Addition/Cyclization Sequences

(2011) Dennis Worgull et al.   CHEMISTRY-A EUROPEAN JOURNAL

Aziridine-Mediated Ligation and Site-Specific Modification of Unprotected Peptides

(2011) Frank Brock Dyer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

4-Isoxazolines: Scaffolds for Organic Synthesis

(2010) Teresa M. V. D. Pinho e Melo   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Highly Diastereoselective Baldwin Rearrangement of Isoxazolines intocis-Acylaziridines

(2010) Eric Gayon et al.   JOURNAL OF ORGANIC CHEMISTRY

Macrocyclization of Linear Peptides Enabled by Amphoteric Molecules

(2010) Ryan Hili et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Enantioselective 1,3-Dipolar Cycloadditions of Nitrones with Propioloylpyrazoles and Acryloylpyrazoles Induced by Chiral π-Cation Catalysts

(2010) Akira Sakakura et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Formal Olefination and Acylaziridination of Imidazolones†

(2010) Xing Dai et al.   ORGANIC LETTERS

4-Isoxazolines and pyrroles from allenoates

(2010) Susana M.M. Lopes et al.   TETRAHEDRON

A Dual Gold-Iron Catalysis for a One-Pot Synthesis of 2,3-Dihydroisoxazoles from Propargylic Alcohols and N-Protected Hydroxylamines

(2009) Olivier Debleds et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic, Enantioselective Ring Opening of Aziridines

(2009) Christoph Schneider   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Aziridine alkaloids as potential therapeutic agents

(2009) Fyaz M.D. Ismail et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

One Pot Synthesis of Optically Active 4-Isoxazolines by Asymmetric Addition of Alkynylzinc Reagents to Nitrones Followed by Cyclization

(2009) Yutaka Ukaji et al.   HETEROCYCLES

Synthesis of stable isoxazolines by [3+2] cycloaddition of oxaziridines with alkynes

(2008) Marilena Fabio et al.   TETRAHEDRON