Sequential Copper-Catalyzed Sonogashira Coupling, Hydroamination and Palladium-Catalyzed Intramolecular Direct Arylation: Synthesis of Azepino-Fused Isoindolinones

Consecutive Sonogashira Coupling and Hydroamination Cyclization for the Synthesis of Isoindolo[1,2-b]quinazolin-10(12H)-ones Catalyzed by CuI/l-Proline

(2017) Jian-Quan Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Phenanthrothiazoles and 1,2-Di(heteroaryl)benzenes through Successive Pd-Catalyzed Direct Arylations

(2017) Xinzhe Shi et al.   JOURNAL OF ORGANIC CHEMISTRY

Integrated Pd-catalyzed cross-coupling strategies for furnishing α-carbolines

(2017) Misayo Sera et al.   TETRAHEDRON

The study of metal-free and palladium-catalysed synthesis of benzochromenes via direct C–H arylation using unactivated aryl benzyl ethers derived from essential oils as raw materials

(2017) Marlyn C. Ortiz Villamizar et al.   Organic Chemistry Frontiers

Synthesis of indole-annulated sulfur heterocycles using copper-catalysed C–N coupling and palladium-catalysed direct arylation

(2016) Ganesh M. Shelke et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-catalyzed tandem Ullmann type C–N coupling and dehydrative cyclization: synthesis of imidazo[1,2-c]quinazolines

(2016) Nitesh K. Nandwana et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Short Synthesis of Sulfur Analogues of Polyaromatic Hydrocarbons through Three Palladium-Catalyzed C–H Bond Arylations

(2016) Wided Hagui et al.   ORGANIC LETTERS

Direct (Hetero)arylation Reactions of (Hetero)arenes as Tools for the Step- and Atom-Economical Synthesis of Biologically Active Unnatural Compounds Including Pharmaceutical Targets

(2016) Renzo Rossi et al.   SYNTHESIS-STUTTGART

Reactivity of 1-(2-bromobenzyl)-4-halopyrazoles in intermolecular and intramolecular Pd-catalysed direct arylations

(2016) Mariem Brahim et al.   TETRAHEDRON

IntermolecularversusIntramolecular Palladium-Catalyzed Direct Arylations between 1-(2-Bromobenzyl)imidazoles and Aryl Bromides

(2015) Xiaowen Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Iterative C−H Bond Arylations: Synthesis of Medium-Size Heterocycles with a Bridgehead Nitrogen Atom

(2015) Wided Hagui et al.   ChemCatChem

Palladium-Catalyzed Synthesis of Phenanthridine/Benzoxazine-Fused Quinazolinones by Intramolecular CH Bond Activation

(2015) Puneet K. Gupta et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Imidazo[1,2-f]phenanthridines through Palladium-Catalyzed Intramolecular C–C Bond Formation

(2015) Anil Kumar et al.   SYNTHESIS-STUTTGART

Cross-Coupling of Heteroarenes by CH Functionalization: Recent Progress towards Direct Arylation and Heteroarylation Reactions Involving Heteroarenes Containing One Heteroatom

(2014) Renzo Rossi et al.   ADVANCED SYNTHESIS & CATALYSIS

Dual Catalysis in DominoN-Benzylation/Intramolecular C-H Arylation: Regio- and Chemoselective Synthesis of Annelated Nitrogen Heterocycles

(2014) Joydev K. Laha et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Aza-Fused Isoquinolines through Domino Cross-Aldol Condensation and Palladium-Catalyzed Intramolecular Direct Arylation

(2014) Shiv Dhiman et al.   JOURNAL OF ORGANIC CHEMISTRY

Modular Synthesis of Benzimidazole-Fused Phenanthridines from 2-Arylbenzimidazoles and o-Dibromoarenes by a Palladium-Catalyzed Cascade Process

(2014) Chunxia Chen et al.   ORGANIC LETTERS

Efficient Synthesis of a (Z)-3-Methyleneisoindolin-1-one Library Using Cu(OAc)2•H2O/DBU under Microwave Irradiation

(2013) Li Zhang et al.   MOLECULES

Direct Functionalization Processes: A Journey from Palladium to Copper to Iron to Nickel to Metal-Free Coupling Reactions

(2012) James J. Mousseau et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of a library of tricyclic azepinoisoindolinones

(2012) Bettina Miller et al.   Beilstein Journal of Organic Chemistry

Blood Pressure in Renal Disease: How to Accomplish the Goal?

(2012) Nicolás R. Robles et al.   Cardiovascular Therapeutics

Synthesis of Fused Imidazoles, Pyrroles, and Indoles with a Defined Stereocenter α to Nitrogen Utilizing Mitsunobu Alkylation Followed by Palladium-Catalyzed Cyclization

(2011) Joydev K. Laha et al.   JOURNAL OF ORGANIC CHEMISTRY

Atroposelective formation of dibenz[c,e]azepines via intramolecular direct arylation with centre-axis chirality transfer

(2011) Caroline A. Cheetham et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthetic Studies on Indolocarbazoles: Total Synthesis of Staurosporine Aglycon

(2011) Ganesan Gobi Rajeshwaran et al.   ORGANIC LETTERS

Importance of palladium–carbon bond energies in direct arylation of polyfluorinated benzenes

(2010) Julie Guihaumé et al.   DALTON TRANSACTIONS

Intramolecular arylation reactions: first efficient synthesis of novel fused pyridoimidazoquinolinones or pyridoimidazoazepinones libraries

(2010) J. Koubachi et al.   TETRAHEDRON

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent advances in aryl–aryl bond formation by direct arylation

(2009) Gerard P. McGlacken et al.   CHEMICAL SOCIETY REVIEWS

Assembly of Substituted 3-Methyleneisoindolin-1-ones via a CuI/l-Proline-Catalyzed Domino Reaction Process of 2-Bromobenzamides and Terminal Alkynes

(2009) Li Li et al.   ORGANIC LETTERS

A New Industrial Process for 10-Methoxyiminostilbene: Key Intermediate for the Synthesis of Oxcarbazepine

(2009) Harnam Singh et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Copper-catalyzed tandem synthesis of [1,2,3]triazolo[5,1-a]isoquinolines and their transformation to 1,3-disubstituted isoquinolines

(2009) Yuan-Yuan Hu et al.   TETRAHEDRON

Generation of novel, potent urotensin-II receptor antagonists by alkylation–cyclization of isoindolinone C3-carbanions

(2009) Diane K. Luci et al.   TETRAHEDRON LETTERS

Pestalachlorides A–C, antifungal metabolites from the plant endophytic fungus Pestalotiopsis adusta

(2008) Erwei Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Intramolecular cyclization reaction — Palladium(0)-catalyzed cyclization is more effective than tin hydride mediated reaction

(2008) Krishna C Majumdar et al.   CANADIAN JOURNAL OF CHEMISTRY

Palladium-mediated synthesis of poly-fused heterocycles from Baylis–Hillman adducts

(2008) Hyun Seung Lee et al.   TETRAHEDRON