Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines

Title
Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines
Authors
Keywords
Pyridylchalcones, Cisplatin-resistance, CYP1B1 inhibitors, Live CYP1B1-Expressing human cells, Live CYP1B1-Expressing yeast cells, Sacchrosomes™
Journal
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 129, Issue -, Pages 159-174
Publisher
Elsevier BV
Online
2017-02-10
DOI
10.1016/j.ejmech.2017.02.016

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