Anti-nociceptive and desensitizing effects of olvanil on capsaicin-induced thermal hyperalgesia in the rat

The contribution of the endogenous TRPV1 ligands 9-HODE and 13-HODE to nociceptive processing and their role in peripheral inflammatory pain mechanisms

(2012) Mohammad Alsalem et al.   BRITISH JOURNAL OF PHARMACOLOGY

Olvanil acts on transient receptor potential vanilloid channel 1 and cannabinoid receptors to modulate neuronal transmission in the trigeminovascular system

(2012) Jan Hoffmann et al.   PAIN

TRPV1 agonist piperine but not olvanil enhances glutamatergic spontaneous excitatory transmission in rat spinal substantia gelatinosa neurons

(2011) Liu Yang et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Topical capsaicin for pain management: therapeutic potential and mechanisms of action of the new high-concentration capsaicin 8% patch

(2011) P. Anand et al.   BRITISH JOURNAL OF ANAESTHESIA

N-palmitoyl-vanillamide (palvanil) is a non-pungent analogue of capsaicin with stronger desensitizing capability against the TRPV1 receptor and anti-hyperalgesic activity

(2011) Luciano De Petrocellis et al.   PHARMACOLOGICAL RESEARCH

Pungency of TRPV1 agonists is directly correlated with kinetics of receptor activation and lipophilicity

(2010) Daniel Ursu et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Therapeutic potential of vanilloid receptor TRPV1 agonists and antagonists as analgesics: Recent advances and setbacks

(2008) Gilbert Y. Wong et al.   BRAIN RESEARCH REVIEWS

Peripheral TRPV1 Receptors As Targets for Drug Development: New Molecules and Mechanisms

(2008) Arpad Szallasi et al.   CURRENT PHARMACEUTICAL DESIGN

HC-030031, a TRPA1 Selective Antagonist, Attenuates Inflammatory- and Neuropathy-Induced Mechanical Hypersensitivity

(2008) Samer R Eid et al.   Molecular Pain

Body-temperature maintenance as the predominant function of the vanilloid receptor TRPV1

(2008) Narender R. Gavva   TRENDS IN PHARMACOLOGICAL SCIENCES