Journal
TETRAHEDRON LETTERS
Volume 57, Issue 14, Pages 1597-1599Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2016.02.102
Keywords
[3+2] cycloaddition; Silver catalysis; Trimethylsilyldiazomethane; 2H-Tetrazole
Categories
Funding
- National Institutes of Health, National Institute on Drug Abuse Grant [P01DA033622]
- [1S10OD010603-01A1]
Ask authors/readers for more resources
A regioselective cycloaddition reaction of arenediazonium salts with trimethylsilyldiazomethane is reported. A series of 2-aryltetrazoles were obtained in good to moderate yields with wide functional group compatibility. Furthermore, this cycloaddition reaction opens the way to build up the versatile intermediate 2-aryl-5-bromotetrazole. (C) 2016 Elsevier Ltd. All rights reserved.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available