PET radiotracer development for imaging high-affinity state of dopamine D2 and D3 receptors: Binding studies of fluorine-18 labeled aminotetralins in rodents

Dopamine D3 receptor binding of18F-fallypride: Evaluation usingin vitroandin vivoPET imaging studies

(2015) Jogeshwar Mukherjee et al.   SYNAPSE

Synthesis and evaluation in rats of homologous series of [18F]-labeled dopamine D2/3 receptor agonists based on the 2-aminomethylchroman scaffold as potential PET tracers

(2015) Vladimir Shalgunov et al.   EJNMMI Research

Convenient synthesis of18F-radiolabeled R-(−)-N-n-propyl-2-(3-fluoropropanoxy-11-hydroxynoraporphine

(2014) Anna W. Sromek et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

18F-MCL-524, an 18F-Labeled Dopamine D2 and D3 Receptor Agonist Sensitive to Dopamine: A Preliminary PET Study

(2014) S. J. Finnema et al.   JOURNAL OF NUCLEAR MEDICINE

Synthesis and Evaluation in Rats of the Dopamine D2/3 Receptor Agonist 18F-AMC20 as a Potential Radioligand for PET

(2014) V. Shalgunov et al.   JOURNAL OF NUCLEAR MEDICINE

Recent methods for measuring dopamine D3 receptor occupancy in vivo: importance for drug development

(2014) Bernard Le Foll et al.   Frontiers in Pharmacology

Heightened D3 Dopamine Receptor Levels in Cocaine Dependence and Contributions to the Addiction Behavioral Phenotype: A Positron Emission Tomography Study with [11C]-(+)-PHNO

(2013) Doris E Payer et al.   NEUROPSYCHOPHARMACOLOGY

Occupancy of Brain Dopamine D3 Receptors and Drug Craving: A Translational Approach

(2012) Manolo Mugnaini et al.   NEUROPSYCHOPHARMACOLOGY

Imaging the high-affinity state of the dopamine D2 receptor in vivo: Fact or fiction?

(2011) Mette Skinbjerg et al.   BIOCHEMICAL PHARMACOLOGY

Within-Subject Comparison of [11C]-( + )-PHNO and [11C]raclopride Sensitivity to Acute Amphetamine Challenge in Healthy Humans

(2011) Paul Shotbolt et al.   JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM

Striatal and extrastriatal microPET imaging of D2/D3 dopamine receptors in rat brain with [18F]fallypride and [18F]desmethoxyfallypride

(2011) Cristian C. Constantinescu et al.   SYNAPSE

All Roads to Schizophrenia Lead to Dopamine Supersensitivity and Elevated Dopamine D2High Receptors

(2010) Philip Seeman   CNS Neuroscience & Therapeutics

Isoflurane Anaesthesia Differentially Affects the Amphetamine Sensitivity of Agonist and Antagonist D2/D3 Positron Emission Tomography Radiotracers: Implications for In Vivo Imaging of Dopamine Release

(2010) Patrick Neil McCormick et al.   MOLECULAR IMAGING AND BIOLOGY

Imaging dopamine receptors in humans with [11C]-(+)-PHNO: Dissection of D3 signal and anatomy

(2010) Andri C. Tziortzi et al.   NEUROIMAGE

Endogenous dopamine (DA) competes with the binding of a radiolabeled D3 receptor partial agonist in vivo: A positron emission tomography study

(2010) Robert H. Mach et al.   SYNAPSE

Performance evaluation of an Inveon PET preclinical scanner

(2009) Cristian C Constantinescu et al.   PHYSICS IN MEDICINE AND BIOLOGY

Dopamine D2/3receptor occupancy of apomorphine in the nonhuman primate brain-A comparative PET study with [11C]raclopride and [11C]MNPA

(2009) Sjoerd J. Finnema et al.   SYNAPSE

In vivo quantification of regional dopamine-D3 receptor binding potential of (+)-PHNO: Studies in non-human primates and transgenic mice

(2009) Eugenii A. Rabiner et al.   SYNAPSE

In vivo 3D digital atlas database of the adult C57BL/6J mouse brain by magnetic resonance microscopy

(2008) Yu Ma   Frontiers in Neuroanatomy