Copper-Catalyzed Direct Sulfoximination of HeteroaromaticN-Oxides by Dual C−H/N−H Dehydrogenative Cross-Coupling

Mechanochemical Rhodium(III)-Catalyzed CH Bond Functionalization of Acetanilides under Solventless Conditions in a Ball Mill

(2015) Gary N. Hermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

[Cp*RhCl2]2: mechanosynthesis and applications in C–H bond functionalisations under ball-milling conditions

(2015) José G. Hernández et al.   CHEMICAL COMMUNICATIONS

Sulfur imidations: access to sulfimides and sulfoximines

(2015) Vincent Bizet et al.   CHEMICAL SOCIETY REVIEWS

Pyridine N-Oxide vs Pyridine Substrates for Rh(III)-Catalyzed Oxidative C–H Bond Functionalization

(2015) Sharon R. Neufeldt et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper(ii)-catalyzed electrophilic amination of quinoline N-oxides with O-benzoyl hydroxylamines

(2015) Gang Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Novel Anthranilic Diamide Insecticides: Design, Synthesis, and Insecticidal Evaluation

(2014) Xuewen Hua et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

Fluorinated sulfoximines: syntheses, properties and applications

(2014) Vincent Bizet et al.   CHEMICAL SOCIETY REVIEWS

Fluorinated Sulfoximines: Preparation, Reactions and Applications

(2014) Xiao Shen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

N-Arylations of Sulfoximines with 2-Arylpyridines by Copper-Mediated Dual N–H/C–H Activation

(2014) Long Wang et al.   ORGANIC LETTERS

Mild Copper–TBAF-Catalyzed N-Arylation of Sulfoximines with Aryl Siloxanes

(2014) Jaeeun Kim et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Amination of Quinoline N-Oxides via C–H Bond Activation under Mild Conditions

(2014) Chongwei Zhu et al.   ORGANIC LETTERS

General synthetic strategies towards N-alkyl sulfoximine building blocks for medicinal chemistry and the use of dimethylsulfoximine as a versatile precursor

(2014) Frederick W. Goldberg et al.   TETRAHEDRON

Palladium-Catalyzed C8-Selective C–H Arylation of Quinoline N-Oxides: Insights into the Electronic, Steric, and Solvation Effects on the Site Selectivity by Mechanistic and DFT Computational Studies

(2014) David E. Stephens et al.   ACS Catalysis

Dimerization of heteroaromatic N-oxides under metal-free conditions

(2014) Hui Wang et al.   RSC Advances

Direct C-2 Alkylation of QuinolineN-Oxides with EthersviaPalladium-Catalyzed Dehydrogenative Cross-Coupling Reaction

(2013) Zhiyong Wu et al.   ADVANCED SYNTHESIS & CATALYSIS

Sulfoximines: A Neglected Opportunity in Medicinal Chemistry

(2013) Ulrich Lücking   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct 2-acetoxylation of quinoline N-oxides via copper catalyzed C–H bond activation

(2013) Xuan Chen et al.   CHEMICAL COMMUNICATIONS

The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor (R)-S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer

(2013) Ulrich Lücking et al.   ChemMedChem

Design, synthesis and biological evaluation of 2-substituted quinolines as potential antileishmanial agents

(2013) Vadiraj S. Gopinath et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Halogenated Quinolines as Substrates for the Palladium-Catalyzed Cross-Coupling Reactions to Afford Substituted Quinolines

(2013) Malose J. Mphahlele et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Copper-Catalyzed Direct Ortho-Alkylation of N-Iminopyridinium Ylides with N-Tosylhydrazones

(2013) Qing Xiao et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Intermolecular Dehydrogenative Amidation/Amination of Quinoline N-Oxides with Lactams/Cyclamines

(2013) Gang Li et al.   ORGANIC LETTERS

Pd-Catalyzed Oxidative CH/CH Direct Coupling of Heterocyclic N-Oxides

(2013) Wei Liu et al.   ORGANIC LETTERS

Sulfonylation of Quinoline N-Oxides with Aryl Sulfonyl Chlorides via Copper-Catalyzed C–H Bonds Activation

(2013) Zhiyong Wu et al.   ORGANIC LETTERS

Sulfoxaflor and the sulfoximine insecticides: Chemistry, mode of action and basis for efficacy on resistant insects

(2013) Thomas C. Sparks et al.   PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY

Copper-Catalyzed Ultrasound-Expedited N-Arylation of Sulfoximines using Diaryliodonium Salts

(2012) Buchireddy Vaddula et al.   ADVANCED SYNTHESIS & CATALYSIS

Syntheses and biological activities of sulfoximine-based acyclic triaryl olefins

(2012) Xiao Yun Chen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Novel diamide insecticides: Sulfoximines, sulfonimidamides and other new sulfonimidoyl derivatives

(2012) Christian Gnamm et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent advances in transition-metal catalyzed reactions using molecular oxygen as the oxidant

(2012) Zhuangzhi Shi et al.   CHEMICAL SOCIETY REVIEWS

N-Cyano Sulfoximines: COX Inhibition, Anticancer Activity, Cellular Toxicity, and Mutagenicity

(2012) Seong Jun Park et al.   ChemMedChem

Origins of regioselectivity of the palladium-catalyzed (aromatic)CH bond metalation–deprotonation

(2012) Serge I. Gorelsky   COORDINATION CHEMISTRY REVIEWS

Transition-State Metal Aryl Bond Stability Determines Regioselectivity in Palladium Acetate Mediated C–H Bond Activation of Heteroarenes

(2012) Alban Petit et al.   ORGANIC LETTERS

The Complementary Competitors: Palladium and Copper in C–N Cross-Coupling Reactions

(2012) Irina P. Beletskaya et al.   ORGANOMETALLICS

Cross-resistance relationships of the sulfoximine insecticide sulfoxaflor with neonicotinoids and other insecticides in the whitefliesBemisia tabaciand Trialeurodes vaporariorum

(2012) Christopher Longhurst et al.   PEST MANAGEMENT SCIENCE

Bioactive sulfoximines: Syntheses and properties of Vioxx® analogs

(2011) Seong Jun Park et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Efficient palladium-catalyzed N-arylation of a sulfoximine with aryl chlorides

(2011) Nattawut Yongpruksa et al.   CHEMICAL COMMUNICATIONS

Palladium-catalyzed desulfitative C-arylation of a benzo[d]oxazole C–H bond with arene sulfonyl chlorides

(2011) Manli Zhang et al.   CHEMICAL COMMUNICATIONS

Quinoline as a Privileged Scaffold in Cancer Drug Discovery

(2011) V. R. Solomon et al.   CURRENT MEDICINAL CHEMISTRY

Palladium-Catalyzed Oxidative Cross-Coupling between PyridineN-Oxides and Indoles

(2011) Xue Gong et al.   ORGANIC LETTERS

Efficient copper-induced coupling between NH-fluoroalkylated sulfoximines and aryl iodides or bromides

(2011) Yohan Macé et al.   TETRAHEDRON

Palladium-Catalyzed Carbonylative CH Activation of Heteroarenes

(2010) Xiao-Feng Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery and Characterization of Sulfoxaflor, a Novel Insecticide Targeting Sap-Feeding Pests

(2010) Yuanming Zhu et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Copper-Catalyzed Direct Sulfoximination of Azoles and Polyfluoroarenes under Ambient Conditions

(2010) Mitsuru Miyasaka et al.   ORGANIC LETTERS

Direct observation of CuI/CuIII redox steps relevant to Ullmann-type coupling reactions

(2010) Alicia Casitas et al.   Chemical Science

Sulfoximine-substituted trifluoromethylpyrimidine analogs as inhibitors of proline-rich tyrosine kinase 2 (PYK2) show reduced hERG activity

(2009) Daniel P. Walker et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Palladium-Catalyzed Alkenylation of Quinoline-N-oxides via C−H Activation under External-Oxidant-Free Conditions

(2009) Junliang Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iron-Catalyzed CN Cross-Coupling of Sulfoximines with Aryl Iodides

(2008) Arkaitz Correa et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed C−H Functionalization of PyridineN-Oxides: Highly Selective Alkenylation and Direct Arylation with Unactivated Arenes

(2008) Seung Hwan Cho et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Analysis of the Concerted Metalation-Deprotonation Mechanism in Palladium-Catalyzed Direct Arylation Across a Broad Range of Aromatic Substrates

(2008) Serge I. Gorelsky et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS