Journal
ORGANIC LETTERS
Volume 18, Issue 9, Pages 2058-2061Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.6b00689
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Funding
- National Basic Research Program of China [2015CB856600]
- National Natural Science Foundation of China [21202184, 21232006, 21572255]
- Chinese Academy of Sciences
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A rhodium(III)-catalyzed cascade cyclization/electrophilic amidation using N-pivaloyloxylamides as the electrophilic nitrogen source has been developed. This protocol provides an efficient route for the synthesis of 3-amidoindoles and 3-amidofurans under mild conditions with good functional group tolerance. The synthetic utility of this reaction has been demonstrated through the derivatization of the 3-amidoindoles to several heterocycle-fused indoles.
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