Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 14, Issue 3, Pages 963-969Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c5ob01915j
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Funding
- Wellcome Trust [WEL081X]
- Cancer Research UK [11566] Funding Source: researchfish
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The one-pot borylation/Suzuki reaction is a very efficient means of accessing cross-coupling products of two aryl-halide partners that generally requires the use of specific catalysts or ligands and/or relatively long reaction times. This new microwave-assisted method provides a quick one-pot borylation/Suzuki reaction protocol that we applied to the synthesis of various bi- or poly-aryl scaffolds, including a variety of aryl and heteroaryl ring systems and the core frameworks of kinase inhibitors vemurafenib and GDC-0879.
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