Optimization and multigram scalability of a catalytic enantioselective borylative migration for the synthesis of functionalized chiral piperidines

Pd-Catalyzed Difluoromethylation of Vinyl Bromides, Triflates, Tosylates, and Nonaflates

(2015) Dalu Chang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric isomerization of allylic alcohols

(2015) Dominique Cahard et al.   TETRAHEDRON LETTERS

Oxygenase-Catalyzed Desymmetrization ofN,N-Dialkyl-piperidine-4-carboxylic Acids

(2014) Anna M. Rydzik et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rings in Drugs

(2014) Richard D. Taylor et al.   JOURNAL OF MEDICINAL CHEMISTRY

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

Regioselective (Diacetoxyiodo)benzene-Promoted Halocyclization of Unfunctionalized Olefins

(2014) Gong-Qing Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of chiral heterocycles by ligand-controlled regiodivergent and enantiospecific Suzuki Miyaura cross-coupling

(2014) Jinyue Ding et al.   Nature Communications

Concise Synthesis and Antimalarial Activity of All Four Mefloquine Stereoisomers Using a Highly Enantioselective Catalytic Borylative Alkene Isomerization

(2013) Jinyue Ding et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Isomerization of Primary Allylic Alcohols into Chiral Aldehydes with the tol-binap/dbapen/Ruthenium(II) Catalyst

(2013) Noriyoshi Arai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Developments in the Synthesis of 1,2-Dihydropyridines

(2013) Artur Silva et al.   SYNTHESIS-STUTTGART

Synthesis of Pyridine and Dihydropyridine Derivatives by Regio- and Stereoselective Addition to N-Activated Pyridines

(2012) James A. Bull et al.   CHEMICAL REVIEWS

Mild Double Allylboration Reactions of Nitriles and Acid Anhydrides Using Potassium Allyltrifluoroborate

(2012) Timothy R. Ramadhar et al.   JOURNAL OF ORGANIC CHEMISTRY

Modified Shapiro Reactions with Bismesitylmagnesium As an Efficient Base Reagent

(2012) William J. Kerr et al.   ORGANIC LETTERS

Intramolecular Pd(II)-Catalyzed Aerobic Oxidative Amination of Alkenes: Synthesis of Six-Membered N-Heterocycles

(2012) Zhan Lu et al.   ORGANIC LETTERS

Carbenylative Amination with N-Tosylhydrazones

(2012) Avinash Khanna et al.   ORGANIC LETTERS

Expanding GSK's solvent selection guide – embedding sustainability into solvent selection starting at medicinal chemistry

(2011) Richard K. Henderson et al.   GREEN CHEMISTRY

Highly Enantioselective Arylation ofN-Tosylalkylaldimines Catalyzed by Rhodium-Diene Complexes

(2011) Zhe Cui et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Targeted drugs by olefin metathesis: piperidine-based iminosugars

(2011) Ileana Dragutan et al.   RSC Advances

FeCl3-Catalyzed Highly Diastereoselective Synthesis of Substituted Piperidines and Tetrahydropyrans

(2010) Amandine Guérinot et al.   ORGANIC LETTERS

Highly enantioselective isomerization of primary allylic alcohols catalyzed by (P,N)-iridium complexes

(2010) Luca Mantilli et al.   PURE AND APPLIED CHEMISTRY

Iridium-Catalyzed Asymmetric Isomerization of Primary Allylic Alcohols

(2009) Luca Mantilli et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

α-Hydroxyalkyl Heterocycles via Chiral Allylic Boronates: Pd-Catalyzed Borylation Leading to a Formal Enantioselective Isomerization of Allylic Ether and Amine

(2009) Stéphanie Lessard et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mild, Rhodium-Catalyzed Intramolecular Hydroamination of Unactivated Terminal and Internal Alkenes with Primary and Secondary Amines

(2008) Zhijian Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of pharmaceutically active compounds containing a disubstituted piperidine framework

(2007) Sara Källström et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Indolizidine and quinolizidine alkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS