Diastereoselective Oxidative CN/CO and CN/CN Bond Formation Tandems Initiated by Visible Light: Synthesis of FusedN-Arylindolines

Intramolecular Dearomative Oxidative Coupling of Indoles: A Unified Strategy for the Total Synthesis of Indoline Alkaloids

(2015) Weiwei Zi et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of Indolines by Copper-Mediated Intramolecular Aromatic C–H Amination

(2015) Kazutaka Takamatsu et al.   JOURNAL OF ORGANIC CHEMISTRY

Concise and Enantioselective Total Synthesis of (−)-Mehranine, (−)-Methylenebismehranine, and RelatedAspidospermaAlkaloids

(2014) Marius Mewald et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Synthesis of [2,3]-Fused Indoline Heterocycles through Inverse-Electron-Demand Aza-Diels-Alder Reaction of Indoles with Azoalkenes

(2014) Min-Chao Tong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(0)-Catalyzed Heck Reaction/CH Activation/Amination Sequence with Diaziridinone: A Facile Approach to Indolines

(2014) Huaiji Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

Metal-Free Protodeboronation of Electron-Rich Arene Boronic Acids and Its Application to ortho-Functionalization of Electron-Rich Arenes Using a Boronic Acid as a Blocking Group

(2014) Su-Jin Ahn et al.   JOURNAL OF ORGANIC CHEMISTRY

Base-Promoted Protodeboronation of 2,6-Disubstituted Arylboronic Acids

(2014) Jerome Lozada et al.   JOURNAL OF ORGANIC CHEMISTRY

Dearomative Indole (3 + 2) Cycloaddition Reactions

(2014) Hui Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of (−)-Pseudotabersonine, (−)-Pseudovincadifformine, and (+)-Coronaridine Enabled by Photoredox Catalysis in Flow

(2014) Joel W. Beatty et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Homogenous Pd-Catalyzed Asymmetric Hydrogenation of Unprotected Indoles: Scope and Mechanistic Studies

(2014) Ying Duan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Visible Light Photoredox Catalysis with Transition Metal Complexes: Applications in Organic Synthesis

(2013) Christopher K. Prier et al.   CHEMICAL REVIEWS

Selection of boron reagents for Suzuki–Miyaura coupling

(2013) Alastair J. J. Lennox et al.   CHEMICAL SOCIETY REVIEWS

Visible-Light-Driven Photoredox Catalysis in the Construction of Carbocyclic and Heterocyclic Ring Systems

(2013) Jun Xuan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Protodeboronation of ortho- and para-Phenol Boronic Acids and Application to ortho and meta Functionalization of Phenols Using Boronic Acids as Blocking and Directing Groups

(2013) Chun-Young Lee et al.   JOURNAL OF ORGANIC CHEMISTRY

Biomedical Importance of Indoles

(2013) Nagendra Kaushik et al.   MOLECULES

Synthesis of Indolines via Pd(II)-Catalyzed Amination of C–H Bonds Using PhI(OAc)2 as the Bystanding Oxidant

(2013) Tian-Sheng Mei et al.   ORGANIC LETTERS

N-Indolyltriethylborate: A Useful Reagent for Synthesis of C3-Quaternary Indolenines

(2013) Aijun Lin et al.   ORGANIC LETTERS

Visible Light Photocatalysis: The Development of Photocatalytic Radical Ion Cycloadditions

(2013) Tehshik P. Yoon   ACS Catalysis

Recent Applications of Organic Dyes as Photoredox Catalysts in Organic Synthesis

(2013) David A. Nicewicz et al.   ACS Catalysis

A Visible-Light-Mediated Oxidative CN Bond Formation/Aromatization Cascade: Photocatalytic Preparation of N-Arylindoles

(2012) Soumitra Maity et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A General Method for Suzuki–Miyaura Coupling Reactions Using Lithium Triisopropyl Borates

(2012) Matthias A. Oberli et al.   ORGANIC LETTERS

Improved Protocol for Indoline Synthesis via Palladium-Catalyzed Intramolecular C(sp2)–H Amination

(2012) Gang He et al.   ORGANIC LETTERS

Synthesis of Oxindolyl Pyrazolines and 3-Amino Oxindole Building Blocks via a Nitrile Imine [3 + 2] Cycloaddition Strategy

(2012) Anand Singh et al.   ORGANIC LETTERS

Rhodium-Catalyzed Synthesis of 2,3-Disubstituted Indoles from β,β-Disubstituted Stryryl Azides

(2011) Ke Sun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Suzuki-Miyaura coupling of heteroaryl boronic acids and vinyl chlorides

(2011) Ashish Thakur et al.   CHEMICAL COMMUNICATIONS

Transmetalation of Unsaturated Carbon Nucleophiles from Boron-Containing Species to the Mid to Late d-Block Metals of Relevance to Catalytic C−X Coupling Reactions (X = C, F, N, O, Pb, S, Se, Te)

(2011) David V. Partyka   CHEMICAL REVIEWS

Structure, Bioactivity and Synthesis of Natural Products with Hexahydropyrrolo[2,3-b]indole

(2011) Pau Ruiz-Sanchis et al.   CHEMISTRY-A EUROPEAN JOURNAL

Heterocycle Synthesis via Direct C–H/N–H Coupling

(2011) Enrico T. Nadres et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Efficient Syntheses of Azetidines, Pyrrolidines, and Indolines via Palladium Catalyzed Intramolecular Amination of C(sp3)–H and C(sp2)–H Bonds at γ and δ Positions

(2011) Gang He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indole synthesis: a review and proposed classification

(2011) Douglass F. Taber et al.   TETRAHEDRON

A New Palladium Precatalyst Allows for the Fast Suzuki−Miyaura Coupling Reactions of Unstable Polyfluorophenyl and 2-Heteroaryl Boronic Acids

(2010) Tom Kinzel et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole

(2010) Simone Lucarini et al.   ORGANIC LETTERS

Gold(I)-Catalyzed Tandem Cyclization Approach to Tetracyclic Indolines

(2010) Yongxiang Liu et al.   ORGANIC LETTERS

Organotrifluoroborates and Monocoordinated Palladium Complexes as Catalysts—A Perfect Combination for Suzuki–Miyaura Coupling

(2009) Gary A. Molander et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

An Interrupted Fischer Indolization Approach toward Fused Indoline-Containing Natural Products

(2009) Ben W. Boal et al.   ORGANIC LETTERS

Palladium-Catalyzed Suzuki−Miyaura Cross-Coupling Reactions Employing Dialkylbiaryl Phosphine Ligands

(2008) Ruben Martin et al.   ACCOUNTS OF CHEMICAL RESEARCH

Dirhodium(II)-Catalyzed Intramolecular CH Amination of Aryl Azides

(2008) Meihua Shen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Scope of the Suzuki−Miyaura Cross-Coupling Reactions of Potassium Heteroaryltrifluoroborates

(2008) Gary A. Molander et al.   JOURNAL OF ORGANIC CHEMISTRY