Synthesis and anti-inflammatory activity of N-arylamides of 4-aryl- and 4-(thiophen-2-yl)-2-[2-(furan-2-carbonyl)hydrazono]-4-oxobutanoic acids

Synthesis of thieno[3,2-e]pyrrolo[1,2-a]pyrimidine derivatives and their precursors containing 2-aminothiophenes fragments as anticancer agents for therapy of pulmonary metastatic melanoma

(2023) Anna Rogova et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Decyclization of Substituted 2-[2-Oxofuran-3(2H)-ylidene)furan-2-carbohydrazides by the Action of Alcohols and Analgesic Activity of the Obtained Compounds

(2023) S. N. Igidov et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Synthesis and Antinociceptive Activity of Substituted 5-(Het)aryl-3-(4-methylbenzoyl)hydrazono-3H-furan-2-ones

(2022) D. V. Lipin et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Synthesis, Intramolecular Cyclization, and Antinociceptive Activity of Substituted 2-[2-(4-Nitrobenzoyl)hydrazinylidene]-4-oxobut-2-enoic Acids

(2022) E. I. Denisova et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Computational-Based Discovery of the Anti-Cancer Activities of Pyrrole-Based Compounds Targeting the Colchicine-Binding Site of Tubulin

(2022) Sergei Boichuk et al.   MOLECULES

Synthesis and anti-inflammatory activity of N′-substituted 2-[2-(diarylmethylene)hydrazinyl]-5,5-dimethyl-4-oxohex-2-enehydrazides

(2022) A. I. Siutkina et al.   RUSSIAN CHEMICAL BULLETIN

Synthesis, analgesic and antimicrobial activity of substituted 2-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-ylamino)-4-oxo-4-phenylbut-2-enoates

(2022) Yu. O. Sharavyeva et al.   RUSSIAN CHEMICAL BULLETIN

Synthesis, Intramolecular Cyclization, and Analgesic Activity of Substituted 2-[2-(Furancarbonyl)hydrazinylydene]-4-oxobutanoic Acids

(2022) S. N. Igidov et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

The Design, Synthesis, and Biological Activities of Pyrrole-Based Carboxamides: The Novel Tubulin Inhibitors Targeting the Colchicine-Binding Site

(2021) Sergei Boichuk et al.   MOLECULES

The influence of substitutes on the room temperature photoluminescence of 2-amino-4-oxobut-2-enoic acid molecular crystals

(2021) Ekaterina Gunina et al.   Photonics and Nanostructures-Fundamentals and Applications

Synthesis and Biological Activity of Substituted 2-[2-(Diphenylmethylene)hydrazinyl]-5,5-dimethyl-4-oxohex-2-enoates

(2021) A. I. Siutkina et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Cytostatic Activity of (E)-Ethyl-2-Amino-5-(3,3-Dimethyl-4-Oxobutyliden)-4-Oxo-1- (2-Phenylaminobenzamido)-4,5-Dihydro-1Hpyrrol-3-Carboxylate

(2020) S. S. Zykova et al.   PHARMACEUTICAL CHEMISTRY JOURNAL

Synthesis, Structure, and Biological Activity of 4-R-4-Oxo-2-[2-(phenylamino)benzoyl]hydrazinylidene-N-hetarylbutanamides

(2020) I. A. Kizimova et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Synthesis of New 2-Aminopyrrole Derivatives by Reaction of Furan-2,3-diones 3-Acylhydrazones with CH-Nucleophiles

(2020) I. A. Kizimova et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Reactions of N'-[2-Oxo-5-R-furan-3(2H)-ylidene]acylhydrazides with Primary and Secondary Alcohols

(2020) I. A. Kizimova et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Synthesis and Biological Activity of N-Aryl(alkyl)-2-[2-(9H-fluoren-9-ylidene)hydrazinylidene]-5,5-dimethyl-4-oxohexanamides

(2019) A. I. Siutkina et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

One-Pot Synthesis of Thieno[3,2-e]pyrrolo[1,2-a]pyrimidine Derivative Scaffold: A Valuable Source of PARP-1 Inhibitors

(2019) Sergei A. Shipilovskikh et al.   JOURNAL OF ORGANIC CHEMISTRY

Chemistry of iminofurans: XIV. Ring opening of 5-substituted furan-2,3-dione 3-benzoylhydrazones by the action of aromatic and heterocyclic amines

(2017) M. A. Kiselev et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Cytotoxic Activity of Ethyl 2-Amino-1-Benzamido-4-Oxo-5-(2-Oxo-2-Arylethylidene)- 4,5-Dihydro-1H-Pyrrole-3-Carboxylates

(2016) S. S. Zykova et al.   PHARMACEUTICAL CHEMISTRY JOURNAL

Synthesis and Pharmacological Activity of Ethyl-2-Amino-1-Benzamido-4-Oxo-5-(2-Oxo-2-Arylethylidene)Pyrrolidine-3-Carboxylates

(2016) S. S. Zykova et al.   PHARMACEUTICAL CHEMISTRY JOURNAL

Synthesis, docking, and biological studies of phenanthrene β-diketo acids as novel HIV-1 integrase inhibitors

(2013) Horrick Sharma et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

SYNTHESIS AND AChE INHIBITING ACTIVITY OF 2, 4 SUBSTITUTED 6-PHENYL PYRIMIDINES

(2013) CRISTIAN PAZ et al.   JOURNAL OF THE CHILEAN CHEMICAL SOCIETY

SYNTHESIS OF THE LIGAND (Z)-2-(3-METHOXYPHENYLAMINO)-4-OXO-4-PHENYLBUT-2-ENOIC ACID AND ITS ANTIFUNGAL ACTIVITY AGAINST THE WOOD STAIN FUNGI MUCOR PLUMBEUS

(2013) C PAZ et al.   JOURNAL OF THE CHILEAN CHEMICAL SOCIETY

Identification of Influenza Endonuclease Inhibitors Using a Novel Fluorescence Polarization Assay

(2012) Brandi M. Baughman et al.   ACS Chemical Biology

Four-Dimensional Structure–Activity Relationship Model to Predict HIV-1 Integrase Strand Transfer Inhibition using LQTA-QSAR Methodology

(2012) Eduardo B. de Melo et al.   Journal of Chemical Information and Modeling

Structural Analysis of Specific Metal Chelating Inhibitor Binding to the Endonuclease Domain of Influenza pH1N1 (2009) Polymerase

(2012) Eva Kowalinski et al.   PLoS Pathogens

A simple and highly efficient preparation of structurally diverse aryl β-diketoacids as hiv-1 integrase inhibitors

(2010) Xiao-Hua Jiang et al.   CHINESE JOURNAL OF CHEMISTRY

Evaluation of HIV-1 integrase inhibitors on human primary macrophages using a luciferase-based single-cycle phenotypic assay

(2010) Zuleika Michelini et al.   JOURNAL OF VIROLOGICAL METHODS

Aryldiketo Acids Have Antibacterial Activity Against MDRStaphylococcus aureusStrains: Structural Insights Based on Similarity and Molecular Interaction Fields

(2009) Branko J. Drakulić et al.   ChemMedChem

The cap-snatching endonuclease of influenza virus polymerase resides in the PA subunit

(2009) Alexandre Dias et al.   NATURE

Targeting Inactive Enzyme Conformation: Aryl Diketoacid Derivatives as a New Class of PTP1B Inhibitors

(2008) Sijiu Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY