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Title
A Selective Cyclic Peptidic Human SIRT5 Inhibitor
Authors
Keywords
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Journal
MOLECULES
Volume 21, Issue 9, Pages 1217
Publisher
MDPI AG
Online
2016-09-12
DOI
10.3390/molecules21091217
References
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Related references
Note: Only part of the references are listed.- Simple N ε -thioacetyl-lysine-containing cyclic peptides exhibiting highly potent sirtuin inhibition
- (2016) Yajun Huang et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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- SIRT5 Regulates both Cytosolic and Mitochondrial Protein Malonylation with Glycolysis as a Major Target
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- Chemical Probing of the Human Sirtuin 5 Active Site Reveals Its Substrate Acyl Specificity and Peptide-Based Inhibitors
- (2014) Claudia Roessler et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Lysine Glutarylation Is a Protein Posttranslational Modification Regulated by SIRT5
- (2014) Minjia Tan et al. Cell Metabolism
- Sirtuins, metabolism, and DNA repair
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- Sirtuin inhibitors as anticancer agents
- (2014) Jing Hu et al. Future Medicinal Chemistry
- Nonenzymatic Protein Acylation as a Carbon Stress Regulated by Sirtuin Deacylases
- (2014) Gregory R. Wagner et al. MOLECULAR CELL
- The growing landscape of lysine acetylation links metabolism and cell signalling
- (2014) Chunaram Choudhary et al. NATURE REVIEWS MOLECULAR CELL BIOLOGY
- SIRT5 Regulates the Mitochondrial Lysine Succinylome and Metabolic Networks
- (2013) Matthew J. Rardin et al. Cell Metabolism
- Activation of the Protein Deacetylase SIRT6 by Long-chain Fatty Acids and Widespread Deacylation by Mammalian Sirtuins
- (2013) Jessica L. Feldman et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Sirtuins in neurodegenerative diseases: an update on potential mechanisms
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- Thiosuccinyl Peptides as Sirt5-Specific Inhibitors
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- Mechanism-based Modulator Discovery for Sirtuin-catalyzed Deacetylation Reaction
- (2012) Weiping Zheng MINI-REVIEWS IN MEDICINAL CHEMISTRY
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- The First Identification of Lysine Malonylation Substrates and Its Regulatory Enzyme
- (2011) Chao Peng et al. MOLECULAR & CELLULAR PROTEOMICS
- Sirt5 Is a NAD-Dependent Protein Lysine Demalonylase and Desuccinylase
- (2011) J. Du et al. SCIENCE
- Distinct regulation of mitochondrial localization and stability of two human Sirt5 isoforms
- (2010) Nobuko Matsushita et al. GENES TO CELLS
- Ten years of NAD-dependent SIR2 family deacetylases: implications for metabolic diseases
- (2010) Shin-ichiro Imai et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- Discovery of potent, proteolytically stable, and cell permeable human sirtuin peptidomimetic inhibitors containing Nε-thioacetyl-lysine
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- Sirtuin/Sir2 phylogeny, evolutionary considerations and structural conservation
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- Role of CYP2E1 in thioacetamide-induced mouse hepatotoxicity
- (2007) Jin Seok Kang et al. TOXICOLOGY AND APPLIED PHARMACOLOGY
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