Radiation Dosimetry of a Novel Adenosine A2A Receptor Radioligand [11C]Preladenant Based on PET/CT Imaging and Ex Vivo Biodistribution in Rats

Synthesis and Preclinical Evaluation of 2-(2-Furanyl)-7-[2-[4-[4-(2-[11C]methoxyethoxy)phenyl]-1-piperazinyl]ethyl]7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine-5-amine ([11C]Preladenant) as a PET Tracer for the Imaging of Cerebral Adenosine A2A Receptors

(2014) Xiaoyun Zhou et al.   JOURNAL OF MEDICINAL CHEMISTRY

Preclinical radiation dosimetry for the novel SV2A radiotracer [18F]UCB-H

(2013) Florian Bretin et al.   EJNMMI Research

Biodistribution and Radiation Dosimetry of the Integrin Marker 18F-RGD-K5 Determined from Whole-Body PET/CT in Monkeys and Humans

(2012) M. Doss et al.   JOURNAL OF NUCLEAR MEDICINE

Evaluation of [18F]Mefway Biodistribution and Dosimetry Based on Whole-Body PET Imaging of Mice

(2012) Cristian C. Constantinescu et al.   MOLECULAR IMAGING AND BIOLOGY

Characterisation of partial volume effect and region-based correction in small animal positron emission tomography (PET) of the rat brain

(2012) Wencke Lehnert et al.   NEUROIMAGE

Suggested pathway to assess radiation safety of 11C-labeled PET tracers for first-in-human studies

(2011) Paolo Zanotti-Fregonara et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

MIRD Pamphlet No. 21: A Generalized Schema for Radiopharmaceutical Dosimetry--Standardization of Nomenclature

(2009) W. E. Bolch et al.   JOURNAL OF NUCLEAR MEDICINE

Human Dosimetry of Carbon-11 Labeled N-butan-2-yl-1-(2-chlorophenyl)-N-methylisoquinoline-3-carboxamide Extrapolated from Whole-body Distribution Kinetics and Radiometabolism in Rats

(2009) Pauliina Luoto et al.   MOLECULAR IMAGING AND BIOLOGY

Potential Therapeutic Interest of Adenosine A2A Receptors in Psychiatric Disorders

(2008) Rodrigo Cunha et al.   CURRENT PHARMACEUTICAL DESIGN

Guideline to regulations for radiopharmaceuticals in early phase clinical trials in the EU

(2008) Alfons Verbruggen et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Radiation Dose Estimates for [18F]5-Fluorouracil Derived from PET-Based and Tissue-Based Methods in Rats

(2008) Adam L. Kesner et al.   MOLECULAR IMAGING AND BIOLOGY