Synthesis of Tetrahydroazepines through Silyl Aza-Prins Cyclization Mediated by Iron(III) Salts

Azetidiniums: Ring-Expansion to Pyrrolidines, Piperidines, Azepanes and Azocanes

(2020) Guillaume Masson et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Structural classification and biological activities of Stemona alkaloids

(2019) Harald Greger   PHYTOCHEMISTRY REVIEWS

1,3-Di- n -butylimidazolium tribromide [BBim]Br 3 : An efficient recyclable catalyst mediated synthesis of N -substituted azepines and their biological evaluation-interaction study with human serum albumin

(2018) Swetha K. Maddili et al.   JOURNAL OF PHOTOCHEMISTRY AND PHOTOBIOLOGY B-BIOLOGY

Synthesis of Various Heterocycles Having a Dienamide Moiety by Ring-Closing Metathesis of Ene-ynamides

(2018) Hideaki Wakamatsu et al.   SYNTHESIS-STUTTGART

Preparation of bicyclic β-lactam and bicyclic 1,3-oxazinone scaffolds using combined cycloaddition and metathesis processes

(2018) Anna Zakaszewska et al.   SYNTHETIC COMMUNICATIONS

Iron-Catalyzed Prins-Peterson Reaction for the Direct Synthesis of Δ4-2,7-disubstituted oxepenes.

(2018) Daniel A Cruz et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric intramolecular Friedel–Crafts reaction catalyzed by a spiro-pyrrolidine organocatalyst: enantioselective construction of indolizine and azepine frameworks

(2018) Yi-Hang Zhang et al.   TETRAHEDRON LETTERS

Synthesis of functionalised azepanes and piperidines from bicyclic halogenated aminocyclopropane derivatives

(2017) Cheng Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A simple and efficient method for constructing azepino[4,5-b]indole derivatives via acid catalysis

(2017) Siva Senthil Kumar Boominathan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

DPPF-Catalyzed Atom-Transfer Radical Cyclization via Allylic Radical

(2017) Longlei Hou et al.   ORGANIC LETTERS

Rhodium(I)-Catalyzed Intermolecular Aza-[4+3] Cycloaddition of Vinyl Aziridines and Dienes: Atom-Economical Synthesis of Enantiomerically Enriched Functionalized Azepines

(2016) Chao-Ze Zhu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantiodivergent Synthesis of (+)- and (−)-Pyrrolidine 197B: Synthesis oftrans-2,5-Disubstituted Pyrrolidines by Intramolecular Hydroamination

(2016) Sixto J. Pérez et al.   CHEMISTRY-A EUROPEAN JOURNAL

Discovery of (R,E)-N-(7-Chloro-1-(1-[4-(dimethylamino)but-2-enoyl]azepan-3-yl)-1H-benzo[d]imidazol-2-yl)-2-methylisonicotinamide (EGF816), a Novel, Potent, and WT Sparing Covalent Inhibitor of Oncogenic (L858R, ex19del) and Resistant (T790M) EGFR Mutants for the Treatment of EGFR Mutant Non-Small-Cell Lung Cancers

(2016) Gérald Lelais et al.   JOURNAL OF MEDICINAL CHEMISTRY

Competitive Ring Expansion of Azetidines into Pyrrolidines and/or Azepanes

(2016) Bruno Drouillat et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Azepane Derivatives by Silyl-aza-Prins Cyclization of Allylsilyl Amines: Influence of the Catalyst in the Outcome of the Reaction

(2016) Asunción Barbero et al.   ORGANIC LETTERS

Enantioselective synthesis of seven-membered carbo- and heterocyles by organocatalyzed intramolecular Michael addition

(2016) James O. Guevara-Pulido et al.   RSC Advances

Stereoselective synthesis of pyrrolidines from β′-amino-allylsilanes

(2015) Peter Mohr et al.   TETRAHEDRON LETTERS

Hexafluoroantimonic Acid Catalysis: Formal [3+2+2] Cycloaddition of Aziridines with Two Alkynes

(2014) Ming-Bo Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

N-Bromosuccinimide-Induced Aminocyclization–Aziridine Ring-Expansion Cascade: An Asymmetric and Highly Stereoselective Approach toward the Synthesis of Azepane

(2014) Jing Zhou et al.   ORGANIC LETTERS

Broadening the Synthetic Scope of the Iron(III)-Catalyzed Aza-Prins Cyclization

(2010) Rubén M. Carballo et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Concise Access to Pyrimidine-Annulated Azepine and Azocine Derivatives by Ruthenium-Catalyzed Ring-Closing Metathesis

(2010) K. Majumdar et al.   SYNTHESIS-STUTTGART

Synthesis of Azepine- and Azocine-Annulated Heterocycles by Aromatic Aza-Claisen Rearrangement and Ring-Closing Metathesis

(2009) K. Majumdar et al.   SYNTHESIS-STUTTGART

A New Catalytic Prins Cyclization Leading to Oxa- and Azacycles

(2008) Pedro O. Miranda et al.   ORGANIC LETTERS