In vivo evaluation of [11C]preladenant positron emission tomography for quantification of adenosine A2A receptors in the rat brain

Characterization in Humans of 18F-MNI-444, a PET Radiotracer for Brain Adenosine 2A Receptors

(2015) O. Barret et al.   JOURNAL OF NUCLEAR MEDICINE

Synthesis and Preclinical Evaluation of 2-(2-Furanyl)-7-[2-[4-[4-(2-[11C]methoxyethoxy)phenyl]-1-piperazinyl]ethyl]7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine-5-amine ([11C]Preladenant) as a PET Tracer for the Imaging of Cerebral Adenosine A2A Receptors

(2014) Xiaoyun Zhou et al.   JOURNAL OF MEDICINAL CHEMISTRY

Development of [18F]-Labeled Pyrazolo[4,3-e]-1,2,4- triazolo[1,5-c]pyrimidine (SCH442416) Analogs for the Imaging of Cerebral Adenosine A2A Receptors with Positron Emission Tomography

(2014) Shivashankar Khanapur et al.   JOURNAL OF MEDICINAL CHEMISTRY

Adenosine 2A Receptor Occupancy by Tozadenant and Preladenant in Rhesus Monkeys

(2014) O. Barret et al.   JOURNAL OF NUCLEAR MEDICINE

Test-retest variability of adenosine A2A binding in the human brain with 11C-TMSX and PET

(2014) Mika Naganawa et al.   EJNMMI Research

Safety, tolerability and pharmacokinetics after single and multiple doses of preladenant (SCH420814) administered in healthy subjects

(2012) D. L. Cutler et al.   JOURNAL OF CLINICAL PHARMACY AND THERAPEUTICS

Adenosine A2A receptors control neuroinflammation and consequent hippocampal neuronal dysfunction

(2011) Nelson Rebola et al.   JOURNAL OF NEUROCHEMISTRY

Adenosine 2A receptor availability in dyskinetic and nondyskinetic patients with Parkinson disease

(2011) A. F. Ramlackhansingh et al.   NEUROLOGY

Adenosine A2A Receptors Measured with [11C]TMSX PET in the Striata of Parkinson's Disease Patients

(2011) Masahiro Mishina et al.   PLoS One

Adenosine A2A Receptors and A2A Receptor Heteromers as Key Players in Striatal Function

(2011) Sergi Ferré et al.   Frontiers in Neuroanatomy

Adenosine receptors and brain diseases: Neuroprotection and neurodegeneration

(2010) Catarina V. Gomes et al.   BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES

Potential Therapeutic Interest of Adenosine A2A Receptors in Psychiatric Disorders

(2008) Rodrigo Cunha et al.   CURRENT PHARMACEUTICAL DESIGN

Positron emission tomography analysis of [11C]KW‐6002 binding to human and rat adenosine A2Areceptors in the brain

(2008) D.J. Brooks et al.   SYNAPSE