Enhancing the Extent of Enolization for α-C–H Bonds of Aliphatic Carboxylic Acid Equivalents via Ion Pair Catalysis: Application toward α-Chalcogenation

Transition Metal‐Free, Free‐Radical Sulfenylation of the α‐C(sp3)‐H Bond in Arylacetamides and Its Application Toward 2‐Thiomethyl Benzoxazoles Synthesis

(2021) Shanghui Tian et al.   ADVANCED SYNTHESIS & CATALYSIS

Functionalization of C(sp3)-H bonds adjacent to heterocycles catalyzed by earth abundant transition metals

(2021) Aniket Gupta et al.   TETRAHEDRON

Catalytic Approaches for the Direct Heterofunctionalization of Aliphatic Carboxylic Acids and Their Equivalents with Group 16 Elements

(2020) Jogendra Kumar et al.   Chemistry-An Asian Journal

Transition Metal‐Free Selective C(sp3)−H Thiolations of Arylacetamide with Substituted Benzenethiol, Aryl Sulfenylchloride and Diaryl Disulfides

(2020) Changying Liu et al.   Asian Journal of Organic Chemistry

Copper-Catalyzed Direct C(sp3)–H Alkoxylation to Access Quaternary α-Alkoxylated Amino Acid Derivatives

(2020) Qiang Wei et al.   ORGANIC LETTERS

Catalytic Direct α-Amination of Arylacetic Acid Synthons with Anilines

(2020) Jogendra Kumar et al.   JOURNAL OF ORGANIC CHEMISTRY

Chemoselective α-Sulfidation of Amides Using Sulfoxide Reagents

(2020) Mario Leypold et al.   ORGANIC LETTERS

α-Fluorination of carbonyls with nucleophilic fluorine

(2019) Pauline Adler et al.   Nature Chemistry

A Chemoselective α-Oxytriflation Enables the Direct Asymmetric Arylation of Amides

(2019) Jing Li et al.   Chem

Direct α-Chalcogenation of Aliphatic Carboxylic Acid Equivalents

(2019) Aniket Gupta et al.   ORGANIC LETTERS

A Mild and Direct C(sp3)–S Cross-Coupling of Oxindoles with Thiols: Synthesis of Unsymmetrical 3-Thiooxindoles

(2019) Hui Qin et al.   JOURNAL OF ORGANIC CHEMISTRY

Unified Approach to the Chemoselective α-Functionalization of Amides with Heteroatom Nucleophiles

(2019) Carlos R. Gonçalves et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Flexible and Chemoselective Oxidation of Amides to α-Keto Amides and α-Hydroxy Amides

(2017) Aurélien de la Torre et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transition-Metal-Free Selective Oxidative C(sp3)–S/Se Coupling of Oxindoles, Tetralone, and Arylacetamides: Synthesis of Unsymmetrical Organochalcogenides

(2017) Ch. Durga Prasad et al.   ORGANIC LETTERS

Chemo- and Stereoselective Transition-Metal-Free Amination of Amides with Azides

(2016) Veronica Tona et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Coordinating activation strategy for C(sp3)–H/C(sp3)–H cross-coupling to access β-aromatic α-amino acids

(2015) Kaizhi Li et al.   Nature Communications

Amino acidic scaffolds bearing unnatural side chains: An old idea generates new and versatile tools for the life sciences

(2014) Andrea Stevenazzi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Development of N-Methyl-(2-arylquinolin-4-yl)oxypropanamides as Leads to PET Radioligands for Translocator Protein (18 kDa)

(2014) Chad Brouwer et al.   JOURNAL OF MEDICINAL CHEMISTRY

Iron-Catalyzed Oxidative CH/CH Cross-Coupling: An Efficient Route to α-Quaternary α-Amino Acid Derivatives

(2013) Kaizhi Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Simple Catalytic Mechanism for the Direct Coupling of α-Carbonyls with Functionalized Amines: A One-Step Synthesis of Plavix

(2013) Ryan W. Evans et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Counteranion-Directed Catalysis: Concept, Definition, and Applications

(2012) Manuel Mahlau et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent Advances in the Synthesis of Unnatural α-Amino Acids - An Updated Version

(2012) A. Perdih et al.   CURRENT ORGANIC CHEMISTRY

Thiol-based angiotensin-converting enzyme 2 inhibitors: P1 modifications for the exploration of the S1 subsite

(2007) David N. Deaton et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS