Fluorine-containing 2,3-diaryl quinolines as potent inhibitors of methicillin and vancomycin-resistant Staphylococcus aureus: Synthesis, antibacterial activity and molecular docking studies

Design, Synthesis, and Dual Evaluation of Quinoline and Quinolinium Iodide Salt Derivatives as Potential Anticancer and Antibacterial Agents

(2020) Guofan Jin et al.   ChemMedChem

C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors

(2020) Tommaso Felicetti et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Discovery of 2-Substituted 3-Arylquinoline Derivatives as Potential Anti-Inflammatory Agents Through Inhibition of LPS-Induced Inflammatory Responses in Macrophages

(2019) Cheng-Yao Yang et al.   MOLECULES

New fluoroquinolones compounds with endo -nortropine derivatives at C-7 position show antibacterial activity against fluoroquinolone-resistant strains of Staphylococcus aureus

(2019) Ramkrushna Ashok Salunke et al.   Chemical Biology & Drug Design

Promising antibacterial agents against multidrug resistant Staphylococcus aureus

(2019) Srikanth Gatadi et al.   BIOORGANIC CHEMISTRY

Halogenated quinolines bearing polar functionality at the 2-position: Identification of new antibacterial agents with enhanced activity against Staphylococcus epidermidis

(2018) Akash Basak et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction

(2018) Tommaso Felicetti et al.   JOURNAL OF MEDICINAL CHEMISTRY

An overview of quinoline as a privileged scaffold in cancer drug discovery

(2017) Robert Musiol   Expert Opinion on Drug Discovery

Metal-Free Synthesis of 2-Substituted 3-(2-Hydroxyaryl)quinolines and 4-(2-Hydroxyaryl)acridines via Benzyne Chemistry

(2017) Ankit Kumar Dhiman et al.   JOURNAL OF ORGANIC CHEMISTRY

Cytotoxicity, antioxidant and antibacterial activity of four compounds produced by an endophytic fungus Epicoccum nigrum associated with Entada abyssinica

(2017) Jean P. Dzoyem et al.   Revista Brasileira de Farmacognosia-Brazilian Journal of Pharmacognosy

Regioselective Metal-Free C2−H Arylation of Quinoline N -Oxides with Aryldiazonium Salts/Anilines under Ambient Conditions

(2017) Rakesh Kumar et al.   Asian Journal of Organic Chemistry

Cytotoxicity, antioxidant and antibacterial activity of four compounds produced by an endophytic fungus Epicoccum nigrum associated with Entada abyssinica

(2017) Jean P. Dzoyem et al.   Revista Brasileira de Farmacognosia-Brazilian Journal of Pharmacognosy

Design, Synthesis and Antibacterial Evaluation of Some New 2-Phenyl-quinoline-4-carboxylic Acid Derivatives

(2016) Xiaoqin Wang et al.   MOLECULES

Comprehensive review on current developments of quinoline-based anticancer agents

(2016) Shweta Jain et al.   Arabian Journal of Chemistry

A novel multiple-stage antimalarial agent that inhibits protein synthesis

(2015) Beatriz Baragaña et al.   NATURE

Treatment of Methicillin-Resistant Staphylococcus aureus: Vancomycin and Beyond

(2015) Natasha Holmes et al.   SEMINARS IN RESPIRATORY AND CRITICAL CARE MEDICINE

Quinoline and quinolones: promising scaffolds for future antimycobacterial agents

(2014) Sandeep Singh et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Novel quinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV

(2013) Mark J. Mitton-Fry et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Methicillin-Resistant Staphylococcus aureus Therapy: Past, Present, and Future

(2013) K. A. Rodvold et al.   CLINICAL INFECTIOUS DISEASES

Medicinal Chemistry of Quinolines As Emerging Anti-inflammatory Agents: An Overview

(2013) S. Mukherjee et al.   CURRENT MEDICINAL CHEMISTRY

Antibiotic resistance—the need for global solutions

(2013) Ramanan Laxminarayan et al.   LANCET INFECTIOUS DISEASES

Emerging Infectious Diseases: Threats to Human Health and Global Stability

(2013) David M. Morens et al.   PLoS Pathogens

Optimization of parameters for semiempirical methods VI: more modifications to the NDDO approximations and re-optimization of parameters

(2012) James J. P. Stewart   JOURNAL OF MOLECULAR MODELING

Quinoline: A versatile heterocyclic

(2012) Akranth Marella et al.   SAUDI PHARMACEUTICAL JOURNAL

Evolution from a Natural Flavones Nucleus to Obtain 2-(4-Propoxyphenyl)quinoline Derivatives As Potent Inhibitors of theS. aureusNorA Efflux Pump

(2011) Stefano Sabatini et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antiproliferative evaluation of 2,3-diarylquinoline derivatives

(2011) Chih-Hua Tseng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Some 2-Aryl- and 2,3-Diaryl-quinolin-4-carboxylic Acid Derivatives

(2011) A. E. M. Saeed et al.   SYNTHETIC COMMUNICATIONS

Serious Infections Caused by Methicillin‐ResistantStaphylococcus aureus

(2010) Helen Boucher et al.   CLINICAL INFECTIOUS DISEASES

Quinolines and structurally related heterocycles as antimalarials

(2010) Kirandeep Kaur et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

(2009) Garrett M. Morris et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY

Infections caused by Gram-positive bacteria: a review of the global challenge

(2009) Neil Woodford et al.   JOURNAL OF INFECTION

Mechanism of Action of the Antibiotic NXL101, a Novel Nonfluoroquinolone Inhibitor of Bacterial Type II Topoisomerases

(2008) M. T. Black et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Synthesis and antibacterial property of quinolines with potent DNA gyrase activity

(2008) Ekambaram Ramesh et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The Many Roles for Fluorine in Medicinal Chemistry

(2008) William K. Hagmann   JOURNAL OF MEDICINAL CHEMISTRY

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS