Design, Synthesis, and Antibacterial Screening of Some Novel Heteroaryl-Based Ciprofloxacin Derivatives as DNA Gyrase and Topoisomerase IV Inhibitors
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Title
Design, Synthesis, and Antibacterial Screening of Some Novel Heteroaryl-Based Ciprofloxacin Derivatives as DNA Gyrase and Topoisomerase IV Inhibitors
Authors
Keywords
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Journal
Pharmaceuticals
Volume 14, Issue 5, Pages 399
Publisher
MDPI AG
Online
2021-04-23
DOI
10.3390/ph14050399
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- (2020) Mohamed Ramadan et al. BIOORGANIC CHEMISTRY
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- (2019) Bahaa G.M. Youssif et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
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- EGFR inhibitors and apoptotic inducers: Design, synthesis, anticancer activity and docking studies of novel xanthine derivatives carrying chalcone moiety as hybrid molecules
- (2019) Hesham A. Abou-Zied et al. BIOORGANIC CHEMISTRY
- Synthesis of imidazole derivatives: Ester and hydrazide compounds with antioxidant activity using ionic liquid as an efficient catalyst
- (2019) Antar A. Abdelhamid et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- Synthesis and characterization of new Cr(III), Fe(III) and Cu(II) complexes incorporating multi-substituted aryl imidazole ligand: Structural, DFT, DNA binding, and biological implications
- (2019) Ahmed M. Abu-Dief et al. SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY
- Synthesis and Evaluation of N -Phenylpyrrolamides as DNA Gyrase B Inhibitors
- (2018) Martina Durcik et al. ChemMedChem
- Current Trends and Future Directions of Fluoroquinolones
- (2018) Hamada H. H. Mohammed et al. CURRENT MEDICINAL CHEMISTRY
- Ciprofloxacin derivatives and their antibacterial activities
- (2018) Gui-Fu Zhang et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- New Method for Synthesis of Multi-substituted Imidazoles
- (2018) Adel A. Marzouk et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- Modifications of quinolones and fluoroquinolones: hybrid compounds and dual-action molecules
- (2018) Joanna Fedorowicz et al. MONATSHEFTE FUR CHEMIE
- Pharmacokinetics and pharmacodynamics of oral pradofloxacin administration in dogs
- (2018) Dawn M. Boothe et al. AMERICAN JOURNAL OF VETERINARY RESEARCH
- Design and Discovery of New Antibacterial Agents: Advances, Perspectives, Challenges
- (2018) Josef Jampilek CURRENT MEDICINAL CHEMISTRY
- Profile of a Novel Anionic Fluoroquinolone—Delafloxacin
- (2018) Paul M Tulkens et al. CLINICAL INFECTIOUS DISEASES
- SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules
- (2017) Antoine Daina et al. Scientific Reports
- Synthesis and anti-mycobacterial activity of 4-(4-phenyl-1H-1,2,3-triazol-1-yl)salicylhydrazones: revitalizing an old drug
- (2016) Hajjaj H. M. Abdu-Allah et al. ARCHIVES OF PHARMACAL RESEARCH
- Design, synthesis and biological evaluation of ciprofloxacin tethered bis-1,2,3-triazole conjugates as potent antibacterial agents
- (2016) Rama Kant et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Conventional and Microwave-assisted Total Synthesis, Antioxidant Capacity, Biological Activity, and Molecular Docking Studies of New Hybrid Compounds
- (2016) Serpil Demirci et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- Synthesis, characterization and biological evaluation of some novel fluoroquinolones
- (2016) Neelanjana Pandit et al. MEDICINAL CHEMISTRY RESEARCH
- Synthesis of novel ciprofloxacin analogues and evaluation of their anti-proliferative effect on human cancer cell lines
- (2013) Narva Suresh et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- New oxadiazole derivatives of isonicotinohydrazide in the search for antimicrobial agents: Synthesis and in vitro evaluation
- (2011) Manav Malhotra et al. JOURNAL OF THE SERBIAN CHEMICAL SOCIETY
- Design, synthesis and biological evaluation of 1,3,4-oxadiazole derivatives
- (2010) Keshari Kishore Jha et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Ciprofloxacin: review on developments in synthetic, analytical, and medicinal aspects
- (2010) Prabodh Chander Sharma et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors ofStaphylococcus aureusMultidrug Efflux Pumps
- (2010) Marco Pieroni et al. JOURNAL OF MEDICINAL CHEMISTRY
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- (2010) Jonathan B. Baell et al. JOURNAL OF MEDICINAL CHEMISTRY
- A roadmap for drug discovery and its translation to small molecule agents in clinical development for tuberculosis treatment
- (2008) H.D. Hollis Showalter et al. TUBERCULOSIS
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