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Synthesis of Novel Pterocarpen Analogues via [3 + 2] Coupling‐Elimination Cascade of α,α‐Dicyanoolefins with Quinone Monoimines

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Identification of potent, selective and orally bioavailable phenyl ((R)-3-phenylpyrrolidin-3-yl)sulfone analogues as RORγt inverse agonists

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(2019) David Marcoux et al.   JOURNAL OF MEDICINAL CHEMISTRY

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Identification of bicyclic hexafluoroisopropyl alcohol sulfonamides as retinoic acid receptor-related orphan receptor gamma (RORγ/RORc) inverse agonists. Employing structure-based drug design to improve pregnane X receptor (PXR) selectivity

(2018) Hua Gong et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Amide-assisted radical strategy: metal-free direct fluorination of arenes in aqueous media

(2017) Deqiang Liang et al.   GREEN CHEMISTRY

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The Emerging Landscape of RORγt Biology

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Highly Enantioselective Hetero-Diels-Alder Reaction of 1,3-Bis(silyloxy)-1,3-dienes with Aldehydes Catalyzed by Chiral Disulfonimide

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(2009) Frank O. Nestle et al.   NEW ENGLAND JOURNAL OF MEDICINE