Antitubercular properties of thiazolidin-4-ones – A review

Synthesis and antimycobacterial activity of thiazolidine-2,4-dione based derivatives with halogenbenzohydrazones and pyridinecarbohydrazones substituents

(2020) Nazar Trotsko et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis and antimycobacterial activity of thiazolidine-2,4-dione-based thiosemicarbazone derivatives

(2020) Nazar Trotsko et al.   BIOORGANIC CHEMISTRY

Synthesis of Novel Sulfamethaoxazole 4-Thiazolidinone Hybrids and Their Biological Evaluation

(2020) Mashooq A. Bhat et al.   MOLECULES

Investigation of (S)-(–)-acidomycin: A selective antimycobacterial natural product that inhibits biotin synthase

(2019) Matthew R Bockman et al.   ACS Infectious Diseases

Dicationic liquid mediated synthesis of tetrazoloquinolinyl methoxy phenyl 4-thiazolidinones and their antibacterial and antitubercular evaluation

(2019) Amarsinh R. Deshmukh et al.   SYNTHETIC COMMUNICATIONS

Influence of Thiazolidine-2,4-Dione Derivatives with Azolidine or Thiosemicarbazone Moieties on Haemophilus spp. Planktonic or Biofilm-Forming Cells

(2019) Nazar Trotsko et al.   MOLECULES

Thiazolidinone/thiazole based hybrids – New class of antitrypanosomal agents

(2019) Anna Kryshchyshyn et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and In Vitro Anti-Toxoplasma gondii Activity of Novel Thiazolidin-4-one Derivatives

(2019) Nazar Trotsko et al.   MOLECULES

Novel thiazolidinedione-hydroxamates as inhibitors of Mycobacterium tuberculosis virulence factor Zmp1

(2019) Veronika Šlachtová et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis, SAR and biological investigation of 3-(carboxymethyl)rhodanine and aminothiazole inhibitors of Mycobacterium tuberculosis Zmp1

(2018) Mattia Mori et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

4-Thiazolidinone coumarin derivatives as two-component NS2B/NS3 DENV flavivirus serine protease inhibitors: synthesis, molecular docking, biological evaluation and structure–activity relationship studies

(2018) Samina Khan Yusufzai et al.   Chemistry Central Journal

Decaprenyl-phosphoryl-ribose 2′-epimerase (DprE1): challenging target for antitubercular drug discovery

(2018) Jineetkumar Gawad et al.   Chemistry Central Journal

Synthesis, in silico molecular docking and pharmacokinetic studies, in vitro antimycobacterial and antimicrobial studies of new imidozolones clubbed with thiazolidinedione

(2018) Imran H. Khan et al.   Current Computer-Aided Drug Design

Synthesis and biological evaluation of 2-aminothiazole-thiazolidinone conjugates as potential antitubercular agents

(2018) Mahmoud F Abo-Ashour et al.   Future Medicinal Chemistry

Design, synthesis and molecular modeling studies of novel thiazolidine-2,4-dione derivatives as potential anti-cancer agents

(2018) Vivek Asati et al.   JOURNAL OF MOLECULAR STRUCTURE

Synthesis and Antibacterial Activity of New Thiazolidine-2,4-dione-Based Chlorophenylthiosemicarbazone Hybrids

(2018) Nazar Trotsko et al.   MOLECULES

Synthesis and antibacterial activity of new (2,4-dioxothiazolidin-5-yl/ylidene)acetic acid derivatives with thiazolidine-2,4-dione, rhodanine and 2-thiohydantoin moieties

(2018) Nazar Trotsko et al.   SAUDI PHARMACEUTICAL JOURNAL

Synthesis and Antibacterial/Antitubercular/Antioxidant Activities of Compounds Containing Fluoroquinolone Ring Linked to a 4-thiazolidinone Moiety

(2018) Tejeswara Rao Allaka et al.   Letters in Drug Design & Discovery

Microwave Assisted, Solvent-Free, “Green” Synthesis of Novel Indole Analogs as Potent Antitubercular and Antimicrobial Agents and Their Molecular Docking Studies

(2018) A. S. Rathod et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Novel indole-thiazolidinone conjugates: Design, synthesis and whole-cell phenotypic evaluation as a novel class of antimicrobial agents

(2018) Mahmoud F. Abo-Ashour et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Quinolidene-rhodanine conjugates: Facile synthesis and biological evaluation

(2017) Dnyaneshwar D. Subhedar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Therapeutic journey of 2,4-thiazolidinediones as a versatile scaffold: An insight into structure activity relationship

(2017) Mohd. Javed Naim et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

5-Ene-4-thiazolidinones – An efficient tool in medicinal chemistry

(2017) Danylo Kaminskyy et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and in vitro antiproliferative and antibacterial activity of new thiazolidine-2,4-dione derivatives

(2017) Nazar Trotsko et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Molecular modeling of drug-pathophysiological Mtb protein targets: Synthesis of some 2-thioxo-1, 3-thiazolidin-4-one derivatives as anti-tubercular agents

(2017) K.M. Noorulla et al.   JOURNAL OF MOLECULAR STRUCTURE

Synthesis and pharmacological studies of 1-(2-amino-1-(4-methoxyphenyl) ethyl) cyclohexanol analogs as potential microbial agents

(2017) Vinay Mahyavanshi et al.   Arabian Journal of Chemistry

Novel tetrazoloquinoline–rhodanine conjugates: Highly efficient synthesis and biological evaluation

(2016) Dnyaneshwar D. Subhedar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and docking studies of pyrazine–thiazolidinone hybrid scaffold targeting dormant tuberculosis

(2016) T.S. Chitre et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Facile synthesis of 1,3-thiazolidin-4-ones as antitubercular agents

(2016) Dnyaneshwar D. Subhedar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design, synthesis and biological screening of new 4-thiazolidinone derivatives with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile

(2016) Khaled R.A. Abdellatif et al.   BIOORGANIC CHEMISTRY

Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives

(2016) Celeste De Monte et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

In Silico Driven Design and Synthesis of Rhodanine Derivatives as Novel Antibacterials Targeting the Enoyl Reductase InhA

(2016) Liudas Slepikas et al.   JOURNAL OF MEDICINAL CHEMISTRY

[Et3NH][HSO4] catalyzed efficient synthesis of 5-arylidene-rhodanine conjugates and their antitubercular activity

(2016) Dnyaneshwar D. Subhedar et al.   RESEARCH ON CHEMICAL INTERMEDIATES

Novel tetrazoloquinoline–thiazolidinone conjugates as possible antitubercular agents: synthesis and molecular docking

(2016) Dnyaneshwar D. Subhedar et al.   MedChemComm

Thiazolidine-2,4-dione derivatives: Programmed chemical weapons for key protein targets of various pathological conditions

(2015) Navriti Chadha et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and Antitubercular activity of New Thiazolidinones with Pyrazinyl and Thiazolyl Scaffolds

(2015) Sambhaji T. Dhumal et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Synthesis of some new 2-amino-6-thiocyanato benzothiazole derivatives bearing 2,4-thiazolidinediones and screening of their in vitro antimicrobial, antitubercular and antiviral activities

(2015) Faiyazalam M. Shaikh et al.   MEDICINAL CHEMISTRY RESEARCH

Synthesis, HIV-1 RT inhibitory, antibacterial, antifungal and binding mode studies of some novel N-substituted 5-benzylidine-2,4-thiazolidinediones

(2015) Radhe Shyam Bahare et al.   DARU-Journal of Pharmaceutical Sciences

New class of methyl tetrazole based hybrid of (Z)-5-benzylidene-2-(piperazin-1-yl)thiazol-4(%H)-one as potent antitubercular agents

(2014) Kuldeep Chauhan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery of the first potent and selective Mycobacterium tuberculosis Zmp1 inhibitor

(2014) Mattia Mori et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Antimycobacterial evaluation of novel hybrid arylidene thiazolidine-2,4-diones

(2014) Singanan Ponnuchamy et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Structure-Guided Design of Thiazolidine Derivatives asMycobacterium tuberculosisPantothenate Synthetase Inhibitors

(2014) Parthiban Brindha Devi et al.   ChemMedChem

Thiazolidine-2,4-diones as multi-targeted scaffold in medicinal chemistry: Potential anticancer agents

(2014) Vivek Asati et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Trends in discovery of new drugs for tuberculosis therapy

(2014) Giovanna Riccardi et al.   JOURNAL OF ANTIBIOTICS

4-Thiazolidinones: The advances continue…

(2013) Avinash C. Tripathi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Structure-Guided Design of Novel Thiazolidine Inhibitors of O-Acetyl Serine Sulfhydrylase from Mycobacterium tuberculosis

(2013) Ömer Poyraz et al.   JOURNAL OF MEDICINAL CHEMISTRY

Novel imidazo[2,1-b][1,3,4]thiadiazole carrying rhodanine-3-acetic acid as potential antitubercular agents

(2012) Shankar G. Alegaon et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Quinoline-based azetidinone and thiazolidinone analogues as antimicrobial and antituberculosis agents

(2012) Bhupendra M. Mistry et al.   MEDICINAL CHEMISTRY RESEARCH

SYNTHESIS OF 4-THIAZOLIDINE DERIVATIVES OF 6-NITROINDAZOLE: PHARMACEUTICAL IMPORTANCE

(2012) PUSHKAL SAMADHIYA et al.   JOURNAL OF THE CHILEAN CHEMICAL SOCIETY

Efficient Regioselective Three-Component Domino Synthesis of 3-(1,2,4-Triazol-5-yl)-1,3-thiazolidin-4-ones as Potent Antifungal and Antituberculosis Agents

(2011) Serry A. El Bialy et al.   ARCHIV DER PHARMAZIE

3,5-Disubstituted-thiazolidine-2,4-dione analogs as anticancer agents: Design, synthesis and biological characterization

(2011) Kai Liu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Low Molecular Weight Phosphotyrosine Protein Phosphatases as Emerging Targets for the Design of Novel Therapeutic Agents

(2011) Rosanna Maccari et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological activity of 4-thiazolidinone derivatives of phenothiazine

(2011) Ritu Sharma et al.   JOURNAL OF THE SERBIAN CHEMICAL SOCIETY

Synthesis and anti-inflammatory activity of new arylidene-thiazolidine-2,4-diones as PPARγ ligands

(2010) Cleiton Diniz Barros et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety

(2010) Dmytro Havrylyuk et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and evaluation of anti-Toxoplasma gondii and antimicrobial activities of thiosemicarbazides, 4-thiazolidinones and 1,3,4-thiadiazoles

(2010) André P. Liesen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of 4-thiazolidinone derivatives as antitubercular and antimicrobial agents

(2010) Pushkal Samadhiya et al.   Arabian Journal of Chemistry

Synthesis and Antimycobacterial Activity of a Novel Series of Isonicotinylhydrazide Derivatives

(2009) Sandip Jaju et al.   ARCHIV DER PHARMAZIE

Synthesis, spectral and biological evaluation of some new thiazolidinones and thiazoles based on t-3-alkyl-r-2,c-6-diarylpiperidin-4-ones

(2009) G. Aridoss et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antibacterial activity of some novel bis-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and bis-4-thiazolidinone derivatives from terephthalic dihydrazide

(2009) Vikrant S. Palekar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of new 4-thiazolidinone derivatives

(2009) Özlen Güzel et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Selective Killing of Nonreplicating Mycobacteria

(2008) Ruslana Bryk et al.   Cell Host & Microbe